SCHEMBL6512897

SCHEMBL6512897

CCCCCOc1ccc(NC(N)=Nc2nc(C)cc(C)n2)cc1F

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 4/20 0.59
RAB9A P51151 3/20 0.59
CRHBP P24387 5/20 0.57
CRHR2 Q13324 5/20 0.57
SMN1; SMN2 Q16637 5/20 0.56
KMT2A Q03164 5/20 0.53
MEN1 O00255 4/20 0.53
CYP1A2 P05177 2/20 0.53
CYP2D6 P10635 2/20 0.53
HCRTR1 O43613 2/20 0.53
CYP2C19 P33261 1/20 0.53
LMNA P02545 3/20 0.50
POLB P06746 2/20 0.50
NPSR1 Q6W5P4 1/20 0.50
MAPT P10636 1/20 0.49
NR4A1 P22736 1/20 0.49
L3MBTL1 Q9Y468 2/20 0.48
ALDH1A1 P00352 1/20 0.48
HTT P42858 2/20 0.47
AHR P35869 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6510787 0.87 MAPK1 (0.56) MAPK1RAB9ACRHBPCRHR2SMN1; SMN2
SCHEMBL5923390 0.78 S1PR1 (0.46) RAB9AKMT2AMAPTALDH1A1
SCHEMBL13338000 0.77 S1PR1 (0.54) MAPT
SCHEMBL4656709 0.77 MAPT (0.64) MAPTALDH1A1
SCHEMBL10637925 0.74 RAB9A (0.54) MAPK1RAB9ACRHBPCRHR2SMN1; SMN2
SCHEMBL9885402 0.73 S1PR1 (0.58) MAPT
SCHEMBL6509463 0.70 CRHBP (0.58) MAPK1RAB9ACRHBPCRHR2KMT2A
SCHEMBL26554065 0.70 S1PR1 (0.58) RAB9ASMN1; SMN2CYP1A2CYP2D6CYP2C19
SCHEMBL28203083 0.70 S1PR1 (0.51) L3MBTL1
SCHEMBL6511099 0.70 CRHBP (0.57) MAPK1RAB9ACRHBPCRHR2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005095345-A2 HETEROARYL GUANIDINES AS INHIBITORS OF VIRAL REPLICATION ACHILLION PHARMACEUTICALS, INC. (US) 2005-10-13 WO claimed