SCHEMBL4657429

SCHEMBL4657429

CC(Cc1ccc(O)c(C(C)(C)C)c1)NC(=O)C(C(C)C)N(C)C(=O)[C@@H](N)Cc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
ALDH1A1 P00352 1/20 0.39
KMT2A Q03164 1/20 0.39
OPRD1 P41143 7/20 0.38
OPRM1 P35372 6/20 0.38
OPRK1 P41145 3/20 0.38
LMNA P02545 1/20 0.38
SLC7A5 Q01650 1/20 0.38
BCHE P06276 4/20 0.37
ACHE P22303 4/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4657436 1.00 NPC1 (0.39) NPC1RAB9AALDH1A1KMT2AOPRD1
SCHEMBL4656090 0.84 CTSS (0.45)
SCHEMBL4656092 0.84 CTSS (0.45)
SCHEMBL4657546 0.83 ABCB1 (0.40) NPC1RAB9AALDH1A1KMT2AOPRD1
SCHEMBL13796438 0.82 MC4R (0.37) NPC1RAB9AKMT2AOPRD1LMNA
SCHEMBL13796434 0.81 MC4R (0.36)
SCHEMBL7947409 0.80 ACACB (0.33) ALDH1A1KMT2AOPRD1OPRM1OPRK1
SCHEMBL13796436 0.80 BACE1 (0.34)
SCHEMBL3989491 0.80 MC4R (0.35) OPRD1OPRM1OPRK1
SCHEMBL3989661 0.80 BACE1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1006122-B1 PHENETHYLAMINE DERIVATIVES CHUGAI PHARMACEUTICAL CO LTD (JP) 2008-12-03 EP claimed
US-6255285-B1 GASTROINTESTINAL DISORDERS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-07-03 US claimed
EP-1006122-A1 PHENETHYLAMINE DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-06-07 EP claimed
EP-1006122-B1 PHENETHYLAMINE DERIVATIVES CHUGAI PHARMACEUTICAL CO LTD (JP) 2008-12-03 EP disclosed
US-6255285-B1 GASTROINTESTINAL DISORDERS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-07-03 US disclosed
EP-1006122-A1 PHENETHYLAMINE DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-06-07 EP disclosed