SCHEMBL4656090

SCHEMBL4656090

CC(Cc1ccc(O)c(C(C)(C)C)c1)NC(=O)C(C(C)C)N(C)C(=O)C(Cc1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSS P25774 8/20 0.45
CTSK P43235 7/20 0.45
CTSB P07858 4/20 0.45
CTSL P07711 2/20 0.45
ACE P12821 1/20 0.44
PTPN1 P18031 2/20 0.42
REN P00797 1/20 0.42
AKT1 P31749 1/20 0.41
KLK5 Q9Y337 1/20 0.40
CA2 P00918 1/20 0.39
HDAC8 Q9BY41 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4656092 1.00 CTSS (0.45) CTSSCTSKCTSBCTSLACE
SCHEMBL4657429 0.84 NPC1 (0.39)
SCHEMBL4657436 0.84 NPC1 (0.39)
SCHEMBL7947409 0.83 ACACB (0.33) CTSSCTSKCTSBPTPN1
SCHEMBL4657546 0.81 ABCB1 (0.40) CTSSCTSKCTSBCTSL
SCHEMBL7947407 0.80 ADRA1A (0.33)
SCHEMBL3989384 0.79 CTSS (0.40) CTSSCTSKCTSBCTSLREN
SCHEMBL3986370 0.79 CTSS (0.40) CTSSCTSKCTSBPTPN1
SCHEMBL3987520 0.77 CTSL (0.41) CTSSCTSKCTSBCTSL
SCHEMBL10657017 0.77 ACE (0.57) CTSSCTSKCTSBCTSLACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1006122-B1 PHENETHYLAMINE DERIVATIVES CHUGAI PHARMACEUTICAL CO LTD (JP) 2008-12-03 EP disclosed
US-6255285-B1 GASTROINTESTINAL DISORDERS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-07-03 US disclosed