SCHEMBL4657463

SCHEMBL4657463

Nc1ccccc1SC(c1ccc(F)cc1)[C@H](NC(=O)OCc1ccccc1)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 0.42
MGLL Q99685 1/20 0.40
CTSL P07711 5/20 0.39
CTSS P25774 5/20 0.39
CTSB P07858 3/20 0.39
CTSK P43235 2/20 0.39
CTRB1 P17538 2/20 0.39
CA2 P00918 2/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA9 Q16790 1/20 0.39
KLK1 P06870 1/20 0.39
ATM Q13315 1/20 0.38
CA5A P35218 1/20 0.38
CNR2 P34972 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4657462 1.00 OPRK1 (0.42) OPRK1MGLLCTSLCTSSCTSB
SCHEMBL5227254 0.93 ATM (0.44) CTSLCTSSCTSBCTSKCTRB1
SCHEMBL5227258 0.93 ATM (0.44) CTSLCTSSCTSBCTSKCTRB1
SCHEMBL3343122 0.92 TRPM8 (0.44) OPRK1MGLLCTSLCTSSCTSB
SCHEMBL3343120 0.92 TRPM8 (0.44) OPRK1MGLLCTSLCTSSCTSB
SCHEMBL5225794 0.91 CTSL (0.39) OPRK1MGLLCTSLCTSSCTSB
SCHEMBL3343179 0.84 TRPM8 (0.48) CTSLCTSSCTSBCTSKATM
SCHEMBL3343181 0.84 TRPM8 (0.48) CTSLCTSSCTSBCTSKATM
SCHEMBL3342679 0.83 TRPM8 (0.44) CTSLCTSSCTSBCTSKCA2
SCHEMBL3550564 0.83 TRPM8 (0.44) CTSLCTSSCTSBCTSKCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1996202-A1 CHEMICAL COMPOUNDS AstraZeneca AB (SE) 2008-12-03 EP disclosed
WO-2007104933-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2007-09-20 WO disclosed