SCHEMBL4658256

SCHEMBL4658256

COc1cccc(OC)c1CNC(=N)N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.43
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
ALDH1A1 P00352 3/20 0.41
ROCK2 O75116 1/20 0.41
PTPN1 P18031 1/20 0.40
KLK1 P06870 1/20 0.40
KLK5 Q9Y337 1/20 0.40
MAPT P10636 2/20 0.40
GAA P10253 1/20 0.40
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
HSD17B10 Q99714 2/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4657734 0.89 KDM1A (0.47) ALDH1A1ROCK2MAPK1
SCHEMBL2380020 0.81 ALDH1A1 (0.39) HIF1AALDH1A1ROCK2PTPN1KLK1
SCHEMBL4018757 0.81 NPSR1 (0.59) ALDH1A1MAPTGAAHDAC1NPSR1
SCHEMBL5735467 0.78 HIF1A (0.40) HIF1AALDH1A1ROCK2PTPN1MAPT
SCHEMBL5723907 0.76 MTNR1A (0.56) HIF1AALDH1A1ROCK2PTPN1NPSR1
SCHEMBL2379469 0.76 HIF1A (0.39) HIF1AALDH1A1ROCK2PTPN1MAPT
SCHEMBL28872280 0.75 HIF1A (0.54) HIF1ACA12CA1CA2CA7
SCHEMBL16950132 0.75 HIF1A (0.49) HIF1ACA12CA1CA2CA4
SCHEMBL1186351 0.74 ALDH1A1 (0.68) CA2ALDH1A1MAPTGAAKDM4E
SCHEMBL28872227 0.74 HIF1A (0.49) HIF1ACA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1917244-A2 HETARYL-SUBSTITUTED GUANIDINE COMPOUNDS AND USE THEREOF AS BINDING PARTNERS FOR 5-HT5-RECEPTORS Abbott GmbH & Co. KG (DE) 2008-05-07 EP disclosed
WO-2007022964-A2 HETARYL-SUBSTITUTED GUANIDINE COMPOUNDS AND USE THEREOF AS BINDING PARTNERS FOR 5-HT5-RECEPTORS ABBOTT GMBH & CO. KG (DE) 2007-03-01 WO disclosed