SCHEMBL4658796

SCHEMBL4658796

COc1cccc(CC(C#N)(C#N)CCC(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.42
IDO1 P14902 2/20 0.42
AGXT P21549 2/20 0.42
CHRM2 P08172 2/20 0.40
CHRM1 P11229 2/20 0.40
CHRM3 P20309 2/20 0.40
PGR P06401 1/20 0.39
AR P10275 1/20 0.39
CMA1 P23946 1/20 0.39
SIGMAR1 Q99720 1/20 0.38
AOC3 Q16853 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
MAOB P27338 1/20 0.38
LPO P22079 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4656238 0.83 MAOB (0.48) MAOB
SCHEMBL4657428 0.82 ALDH1A1 (0.39) TAAR1IDO1AGXTPGRAR
SCHEMBL4657615 0.81 TAAR1 (0.38) TAAR1IDO1ARMEN1KMT2A
SCHEMBL4657339 0.80 TAAR1 (0.39) TAAR1IDO1AGXTCHRM2MAOB
SCHEMBL6821384 0.79 TAAR1 (0.43) TAAR1IDO1AGXTCHRM2CHRM1
SCHEMBL22827424 0.78 TAAR1 (0.55) TAAR1IDO1AGXTCHRM2CHRM1
SCHEMBL4656615 0.78 PNMT (0.40) TAAR1IDO1AGXTMEN1KMT2A
SCHEMBL4656626 0.78 TAAR1 (0.45) TAAR1IDO1SIGMAR1MEN1KMT2A
SCHEMBL4657447 0.77 ATM (0.40) TAAR1
SCHEMBL11089013 0.73 TAAR1 (0.46) TAAR1IDO1AGXTCHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1385817-B1 MALONONITRILE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL CO (JP) 2008-12-03 EP disclosed
US-7402691-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2008-07-22 US disclosed
US-7011838-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2006-03-14 US disclosed
US-20050209323-A1 Malononitrile compounds and their use as pesticides OTAKA KEN 2005-09-22 US disclosed
US-20040138065-A1 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2004-07-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050209323-A1 Malononitrile compounds and their use as pesticides C1S, C1R, C5 TAAR1 644/4885IDO1 382/4885AGXT 510/4885
US-20040138065-A1 Malononitrile compounds and their use as pesticides CBR1, MAL2, CBR3 TAAR1 632/4885IDO1 278/4885AGXT 1757/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.