SCHEMBL4657339

SCHEMBL4657339

N#CC(C#N)(CCC(F)(F)F)Cc1cccc(F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.39
ATM Q13315 1/20 0.38
MIF P14174 1/20 0.38
IDO1 P14902 2/20 0.38
AGXT P21549 2/20 0.38
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 2/20 0.37
PKM P14618 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37
MAOB P27338 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.34
LMNA P02545 2/20 0.34
HTT P42858 2/20 0.34
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
USP2 O75604 1/20 0.34
POLB P06746 1/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4657521 0.83 IDO1 (0.31) IDO1
SCHEMBL4657615 0.83 TAAR1 (0.38) TAAR1ATMIDO1KDM4EMAOB
SCHEMBL4656615 0.83 PNMT (0.40) TAAR1ATMIDO1AGXTALDH1A1
SCHEMBL4656626 0.83 TAAR1 (0.45) TAAR1ATMMIFIDO1ALDH1A1
SCHEMBL4657447 0.82 ATM (0.40) TAAR1ATMALDH1A1SMN1; SMN2LMNA
SCHEMBL4658834 0.80 MAOA (0.33) TAAR1MIFIDO1AGXTALDH1A1
SCHEMBL4658796 0.80 TAAR1 (0.42) TAAR1IDO1AGXTMAOBCHRM2
SCHEMBL4657487 0.79 ALDH1A1 (0.33) ALDH1A1HTT
SCHEMBL4656238 0.76 MAOB (0.48) MAOB
SCHEMBL3647842 0.75 TAAR1 (0.52) TAAR1MIFIDO1AGXTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1385817-B1 MALONONITRILE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL CO (JP) 2008-12-03 EP disclosed
US-7402691-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2008-07-22 US disclosed
US-7011838-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2006-03-14 US disclosed
US-20050209323-A1 Malononitrile compounds and their use as pesticides OTAKA KEN 2005-09-22 US disclosed
US-20040138065-A1 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2004-07-15 US disclosed
EP-1385817-A2 MALONONITRILE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2004-02-04 EP disclosed
WO-2002090320-A2 MALONONITRILE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2002-11-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050209323-A1 Malononitrile compounds and their use as pesticides C1S, C1R, C5 TAAR1 644/4885ATM 4583/4885MIF 898/4885
US-20040138065-A1 Malononitrile compounds and their use as pesticides CBR1, MAL2, CBR3 TAAR1 632/4885ATM 4737/4885MIF 894/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.