SCHEMBL4658917

SCHEMBL4658917

N#CC(C#N)(CCC(F)(F)F)Cc1ccc([N+](=O)[O-])cc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 1/20 0.43
HSD17B10 Q99714 1/20 0.42
KMT2A Q03164 4/20 0.36
TRPV1 Q8NER1 1/20 0.35
PDE7A Q13946 3/20 0.35
MAPT P10636 2/20 0.35
MEN1 O00255 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HSD11B1 P28845 1/20 0.35
LMNA P02545 1/20 0.35
PDK1 Q15118 1/20 0.34
PDK2 Q15119 1/20 0.34
PDK3 Q15120 1/20 0.34
PDK4 Q16654 1/20 0.34
NPC1 O15118 1/20 0.34
MAPK1 P28482 1/20 0.34
RAB9A P51151 1/20 0.34
CRHBP P24387 1/20 0.34
CRHR2 Q13324 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27819708 0.81 HSD17B10 (0.55) VCAM1HSD17B10KMT2ATRPV1PDE7A
SCHEMBL4658455 0.80 GGPS1 (0.42) KMT2AMEN1NPC1MAPK1RAB9A
SCHEMBL4657362 0.79 NR3C1 (0.37) HSD17B10KMT2AMAPTMEN1ALDH1A1
SCHEMBL4657431 0.79 CYP2C19 (0.42) ALDH1A1
SCHEMBL4714787 0.78 MRGPRX4 (0.41) MAPTALDH1A1
SCHEMBL4657492 0.74 IDO1 (0.36) ALDH1A1HSD11B1LMNA
SCHEMBL11566206 0.73 HSD17B10 (0.56) VCAM1HSD17B10KMT2APDE7AMAPT
SCHEMBL30127086 0.72 HSD17B10 (0.55) VCAM1HSD17B10KMT2APDE7AMAPT
SCHEMBL2816576 0.72 HSD17B10 (0.55) VCAM1HSD17B10KMT2APDE7AMAPT
SCHEMBL3710161 0.70 HSD17B10 (0.60) VCAM1HSD17B10KMT2APDE7AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1385817-B1 MALONONITRILE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL CO (JP) 2008-12-03 EP disclosed
US-7402691-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2008-07-22 US disclosed
US-7011838-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2006-03-14 US disclosed
US-20050209323-A1 Malononitrile compounds and their use as pesticides OTAKA KEN 2005-09-22 US disclosed
US-20040138065-A1 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2004-07-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050209323-A1 Malononitrile compounds and their use as pesticides C1S, C1R, C5 VCAM1 4687/4885HSD17B10 1209/4885KMT2A 3658/4885
US-20040138065-A1 Malononitrile compounds and their use as pesticides CBR1, MAL2, CBR3 VCAM1 3383/4885HSD17B10 847/4885KMT2A 2762/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.