SCHEMBL4657362

SCHEMBL4657362

N#CC(C#N)(CCC(F)(F)F)Cc1ccc(F)cc1Cl

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 4/20 0.37
PGR P06401 3/20 0.37
NR3C2 P08235 3/20 0.37
P2RX7 Q99572 5/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 2/20 0.34
HTT P42858 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CYP1A2 P05177 2/20 0.32
CYP2C19 P33261 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
ALOX15 P16050 1/20 0.32
CRHBP P24387 1/20 0.32
CRHR2 Q13324 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4658455 0.87 GGPS1 (0.42) NR3C1PGRNR3C2SMN1; SMN2KDM4E
SCHEMBL4657490 0.85 IDO1 (0.38) NR3C1PGRNR3C2SMN1; SMN2KDM4E
SCHEMBL4714787 0.84 MRGPRX4 (0.41) SMN1; SMN2ALDH1A1KDM4EHTTMAPT
SCHEMBL4657492 0.80 IDO1 (0.36) PGRALDH1A1KDM4E
SCHEMBL4658917 0.79 VCAM1 (0.43) ALDH1A1MAPTTDP1NPC1RAB9A
SCHEMBL4658834 0.74 MAOA (0.33) ALDH1A1KDM4ERAB9AHSD17B10KMT2A
SCHEMBL4657339 0.73 TAAR1 (0.39) SMN1; SMN2ALDH1A1KDM4EHTTMAPT
SCHEMBL4716546 0.73 FDPS (0.40) SMN1; SMN2GAAALOX15SLC6A2SLC6A4
SCHEMBL4657455 0.72 TAAR1 (0.36) NR3C1NR3C2ALDH1A1HTTMAPT
SCHEMBL4657521 0.71 IDO1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1385817-B1 MALONONITRILE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL CO (JP) 2008-12-03 EP disclosed
US-7402691-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2008-07-22 US disclosed
US-7011838-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2006-03-14 US disclosed
US-20050209323-A1 Malononitrile compounds and their use as pesticides OTAKA KEN 2005-09-22 US disclosed
US-20040138065-A1 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2004-07-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050209323-A1 Malononitrile compounds and their use as pesticides C1S, C1R, C5 NR3C1 2356/4885PGR 3230/4885NR3C2 1612/4885
US-20040138065-A1 Malononitrile compounds and their use as pesticides CBR1, MAL2, CBR3 NR3C1 906/4885PGR 4395/4885NR3C2 1214/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.