SCHEMBL4714787

SCHEMBL4714787

N#CC(C#N)(CCC(F)(F)F)Cc1ccc(C(F)(F)F)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 7/20 0.41
DAO P14920 1/20 0.39
ALDH1A1 P00352 2/20 0.37
MAPT P10636 1/20 0.37
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PDE2A O00408 1/20 0.35
HTR2A P28223 4/20 0.34
SLC6A4 P31645 4/20 0.34
KCNH2 Q12809 4/20 0.34
KDM4E B2RXH2 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
AR P10275 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4658455 0.85 GGPS1 (0.42) HTTSMN1; SMN2KDM4EL3MBTL1
SCHEMBL6824476 0.85 MRGPRX4 (0.39) MRGPRX4DAOALDH1A1MAPTHTT
SCHEMBL4657362 0.84 NR3C1 (0.37) ALDH1A1MAPTHTTSMN1; SMN2SLC6A4
SCHEMBL6835194 0.83 MRGPRX4 (0.41) MRGPRX4DAOALDH1A1MAPTHTT
SCHEMBL5007979 0.83 MRGPRX4 (0.40) MRGPRX4DAOALDH1A1MAPTHTT
SCHEMBL4656186 0.81 GABRP (0.33) MRGPRX4ALDH1A1MAPTHTTL3MBTL1
SCHEMBL4657492 0.79 IDO1 (0.36) ALDH1A1KDM4E
SCHEMBL4658917 0.78 VCAM1 (0.43) ALDH1A1MAPT
SCHEMBL4657451 0.75 TAAR1 (0.39) DAOALDH1A1KDM4E
SCHEMBL4656626 0.74 TAAR1 (0.45) ALDH1A1MAPTHTR2ASLC6A4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1385817-B1 MALONONITRILE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL CO (JP) 2008-12-03 EP disclosed
US-7402691-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2008-07-22 US disclosed
US-7011838-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2006-03-14 US disclosed
US-20050209323-A1 Malononitrile compounds and their use as pesticides OTAKA KEN 2005-09-22 US disclosed
US-20040138065-A1 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2004-07-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050209323-A1 Malononitrile compounds and their use as pesticides C1S, C1R, C5 MRGPRX4 430/4885DAO 2284/4885ALDH1A1 1502/4885
US-20040138065-A1 Malononitrile compounds and their use as pesticides CBR1, MAL2, CBR3 MRGPRX4 1431/4885DAO 2052/4885ALDH1A1 614/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.