SCHEMBL4659017

SCHEMBL4659017

CCCC[Sn](CCCC)(CCCC)c1c[nH]c(-c2nc(C)cc(-c3ccc(Cl)c(C)c3)n2)n1

nearest known ligand 0.31

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.31
GRM2 Q14416 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4659002 0.93 KMO (0.34)
SCHEMBL4658975 0.89 CTRC (0.38)
SCHEMBL4660466 0.82 CTSS (0.37)
SCHEMBL4659140 0.78 PTGS2 (0.37)
SCHEMBL4657837 0.76 PTGS2 (0.37)
SCHEMBL4657860 0.76 ABL1 (0.36) ABL1GRM2
SCHEMBL4658258 0.75 KDM4E (0.44)
SCHEMBL3563031 0.74 GRM5 (0.31) GRM2
SCHEMBL4659004 0.72 KDM4E (0.43)
SCHEMBL4657757 0.72 PTGS2 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001849-A1 PYRIDINE AND PYRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS F. Hoffmann-Roche AG (CH) 2008-12-17 EP disclosed
WO-2007110337-A1 PYRIDINE AND PYRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2007-10-04 WO disclosed