SCHEMBL4660256

SCHEMBL4660256

C=C(C(=O)O)c1c2ccccc2nc2ccc(C#N)cc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.44
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 3/20 0.41
PIN1 Q13526 1/20 0.41
MEN1 O00255 5/20 0.40
KMT2A Q03164 5/20 0.40
ATM Q13315 1/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
ADORA2A P29274 1/20 0.39
MAPK1 P28482 2/20 0.38
PKM P14618 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
ABCG2 Q9UNQ0 2/20 0.37
ABCB1 P08183 1/20 0.37
MAPT P10636 2/20 0.37
RAB9A P51151 1/20 0.37
CYP1A2 P05177 4/20 0.36
CYP3A4 P08684 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9330478 0.86 PIN1 (0.48) KDM1AALDH1A1KDM4EPIN1MEN1
SCHEMBL2818996 0.82 PDE10A (0.49) ALDH1A1KDM4EMEN1KMT2AATM
SCHEMBL4660259 0.72 KDM1A (0.43) KDM1AALDH1A1KDM4EPIN1MEN1
SCHEMBL5957199 0.69 ALDH1A1 (0.64) ALDH1A1KDM4EMEN1KMT2ARXFP1
SCHEMBL29392214 0.69 NQO2 (0.50) KDM1AALDH1A1KDM4EPIN1MEN1
SCHEMBL1996329 0.69 NQO2 (0.50) KDM1AALDH1A1KDM4EPIN1MEN1
Water SCHEMBL2991911 0.67 PDE10A (0.63) ALDH1A1KDM4EMEN1KMT2ASMN1; SMN2
SCHEMBL9682802 0.66 KMT2A (0.51) KDM1AALDH1A1KDM4EMEN1KMT2A
SCHEMBL17742243 0.66 ALDH1A1 (0.61) KDM1AALDH1A1KDM4EMEN1KMT2A
SCHEMBL8875118 0.66 SMN1; SMN2 (0.41) ALDH1A1KDM4EMEN1KMT2AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2004628-A2 ACRIDINE DERIVATIVES WITH ANTITUMORAL ACTIVITY Universidade Federal de Pernambuco-Ufpe (BR) 2008-12-24 EP disclosed
WO-2007109871-A2 ACRIDINE DERIVATIVES WITH ANTITUMORAL ACTIVITY UNIVERSIDADE FEDERAL DE PERNAMBUCO - UFPE (BR) 2007-10-04 WO disclosed