SCHEMBL4660558

SCHEMBL4660558

C/C(=C/F)Cc1cc(F)cc(F)c1F

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 8/20 0.41
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
TRPA1 O75762 1/20 0.33
NTRK1 P04629 1/20 0.31
CHRM4 P08173 1/20 0.30
ROCK2 O75116 1/20 0.30
ROCK1 Q13464 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4659435 0.78 IDO1 (0.43) RIPK1
SCHEMBL4659409 0.78 MAPK8 (0.40) RIPK1CES2CES1TRPA1
SCHEMBL29517836 0.77 RIPK1 (0.50) RIPK1CES2CES1NTRK1CHRM4
SCHEMBL15271780 0.77 RIPK1 (0.50) RIPK1CES2CES1NTRK1CHRM4
SCHEMBL1294867 0.75 AOC2 (0.40) RIPK1CES2CES1
SCHEMBL1294869 0.75 AOC2 (0.40) RIPK1CES2CES1
SCHEMBL1295619 0.75 AOC2 (0.40) RIPK1CES2CES1
SCHEMBL4660728 0.75 TRPA1 (0.39) RIPK1CES2CES1TRPA1
SCHEMBL6858266 0.72 RIPK1 (0.49) RIPK1CES2CES1NTRK1
SCHEMBL12108023 0.71 RIPK1 (0.39) RIPK1CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2004166-A2 INHIBITORS OF SEMICARBAZIDE-SENSITIVE AMINE OXIDASE (SSAO) AND VAP-1 MEDIATED ADHESION USEFUL FOR TREATMENT AND PREVENTION OF DISEASES LA JOLLA PHARMACEUTICAL COMPANY (US) 2008-12-24 EP claimed
WO-2007120528-A2 INHIBITORS OF SEMICARBAZIDE-SENSITIVE AMINE OXIDASE (SSAO) AND VAP-1 MEDIATED ADHESION USEFUL FOR TREATMENT AND PREVENTION OF DISEASES LA JOLLA PHARMACEUTICAL COMPANY (US) 2007-10-25 WO claimed