SCHEMBL4660559

SCHEMBL4660559

CC(=O)CC(N)C(=O)O.O=S(=O)(O)c1ccccc1

nearest known ligand 0.52

Known targets — ChEMBL curated mechanism

BTKCACNA1CCACNA1DCACNA1FCACNA1SCACNA2D1CACNA2D2DRD2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQHRH1HTR2AP2RY12

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
ALPI P09923 1/20 0.47
PKM P14618 1/20 0.47
PTGS1 P23219 1/20 0.47
XIAP P98170 1/20 0.47
SLC7A5 Q01650 1/20 0.47
CASR P41180 4/20 0.46
GRIK1 P39086 2/20 0.44
GRIK2 Q13002 1/20 0.44
LARS1 Q9P2J5 1/20 0.42
KYNU Q16719 2/20 0.42
SLC1A3 P43003 2/20 0.41
SLC1A2 P43004 2/20 0.41
SLC1A1 P43005 2/20 0.41
GRM2 Q14416 1/20 0.41
GRM3 Q14832 1/20 0.41
KIF11 P52732 2/20 0.40
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Aspartic Acid SCHEMBL538085 0.87 TSHR (0.55) TSHRSMN1; SMN2ALPIPKMPTGS1
Aspartic Acid SCHEMBL538084 0.87 TSHR (0.55) TSHRSMN1; SMN2ALPIPKMPTGS1
Leucine SCHEMBL11803673 0.84 LARS1 (0.60) TSHRSMN1; SMN2ALPIPKMPTGS1
Leucine SCHEMBL11024352 0.84 LARS1 (0.60) TSHRSMN1; SMN2ALPIPKMPTGS1
Dl-Phenylalanine SCHEMBL25434213 0.82 SLC7A5 (0.73) TSHRSMN1; SMN2ALPIPKMPTGS1
Phenylalanine SCHEMBL25434211 0.82 SLC7A5 (0.73) TSHRSMN1; SMN2ALPIPKMPTGS1
Aspartic Acid SCHEMBL28088617 0.80 TSHR (0.47) TSHRSMN1; SMN2ALPIPKMPTGS1
Alanine SCHEMBL10627958 0.79 TSHR (0.64) TSHRSMN1; SMN2CASRLARS1SLC1A3
Alanine SCHEMBL10626231 0.79 TSHR (0.64) TSHRSMN1; SMN2CASRLARS1SLC1A3
Aspartic Acid SCHEMBL9386444 0.78 TSHR (0.44) TSHRSMN1; SMN2ALPIPKMPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007711-A1 5-AMINOLEVULINIC ACID SALTS AND THEIR USE Bar Ilan University (IL) 2008-12-31 EP disclosed
WO-2007107998-A1 5-AMINOLEVULINIC ACID SALTS AND THEIR USE BAR ILAN UNIVERSITY (IL) 2007-09-27 WO disclosed