SCHEMBL4665305

SCHEMBL4665305

C1=CC(c2nnco2)=N[N]1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 14/20 0.44
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
LMNA P02545 2/20 0.37
TLR8 Q9NR97 1/20 0.37
MAPT P10636 1/20 0.37
HTT P42858 1/20 0.37
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.36
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12906161 0.71 NOTUM (0.59) NOTUMKDM4EALDH1A1LMNATLR8
SCHEMBL17694561 0.67 NOTUM (0.78) NOTUMKDM4EALDH1A1LMNATLR8
SCHEMBL9466191 0.67 LTA4H (0.37)
SCHEMBL2610163 0.66 NOTUM (0.75) NOTUMKDM4EALDH1A1LMNATLR8
SCHEMBL9465018 0.62 KEAP1 (0.43) NOTUMKDM4EALDH1A1LMNA
SCHEMBL9464697 0.62
Methane SCHEMBL28273359 0.60 NOTUM (0.96) NOTUMKDM4EALDH1A1LMNATLR8
SCHEMBL5571187 0.60 NOTUM (0.91) NOTUMKDM4EALDH1A1LMNATLR8
SCHEMBL3685411 0.60 NOTUM (0.64) NOTUMKDM4EALDH1A1LMNATLR8
SCHEMBL14814390 0.60 NOTUM (1.00) NOTUMKDM4EALDH1A1LMNATLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007753-A1 HETEROCYCLIC GABA ALPHA SUBTYPE SELECTIVE RECEPTOR MODULATORS F. Hoffmann-Roche AG (CH) 2008-12-31 EP claimed
WO-2007115966-A1 HETEROCYCLIC GABA ALPHA SUBTYPE SELECTIVE RECEPTOR MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2007-10-18 WO claimed
EP-2007753-A1 HETEROCYCLIC GABA ALPHA SUBTYPE SELECTIVE RECEPTOR MODULATORS F. Hoffmann-Roche AG (CH) 2008-12-31 EP disclosed
WO-2007115966-A1 HETEROCYCLIC GABA ALPHA SUBTYPE SELECTIVE RECEPTOR MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2007-10-18 WO disclosed