SCHEMBL4666768

SCHEMBL4666768

Cc1cc(Nc2ccc(Cl)cc2C(=O)O)n(-c2cnccc2C)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.45
GFER P55789 1/20 0.44
JAK2 O60674 3/20 0.44
JAK1 P23458 3/20 0.44
TYK2 P29597 3/20 0.44
JAK3 P52333 3/20 0.44
KDM4C Q9H3R0 2/20 0.43
MAPT P10636 2/20 0.42
DHODH Q02127 2/20 0.42
LMNA P02545 3/20 0.41
KDM4E B2RXH2 1/20 0.41
HSD17B10 Q99714 1/20 0.41
FTO Q9C0B1 1/20 0.41
NTRK1 P04629 1/20 0.41
GAA P10253 3/20 0.40
HPGD P15428 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
ALPG P10696 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MYC P01106 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4793978 0.89 DHODH (0.47) ADORA1GFERKDM4CMAPTDHODH
SCHEMBL4667612 0.88 GFER (0.44) ADORA1GFERKDM4CMAPTDHODH
SCHEMBL4667080 0.86 GFER (0.57) ADORA1GFERKDM4CMAPTLMNA
SCHEMBL4664665 0.79 TGFBR1 (0.40) ADORA1KDM4CHPGDALDH1A1TGFBR1
SCHEMBL14600184 0.75 ADORA1 (0.49) ADORA1GFERKDM4CMAPTLMNA
SCHEMBL4667046 0.74 ADORA1 (0.52) ADORA1KDM4C
SCHEMBL14600217 0.74 MAPK14 (0.50) ADORA1GFERMAPT
SCHEMBL14600443 0.72 MAPK14 (0.53) JAK2GAA
SCHEMBL8354329 0.71 GFER (0.49) ADORA1GFERJAK2JAK1TYK2
SCHEMBL14600210 0.71 DHODH (0.45) ADORA1KDM4CMAPTDHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928455-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES Bayer Healthcare, LLC (US) 2008-06-11 EP disclosed
WO-2007027842-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES BAYER HEALTHCARE LLC (US) 2007-03-08 WO disclosed
WO-2007027842-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES BAYER HEALTHCARE LLC (US) 2007-03-08 WO disclosed