SCHEMBL4667859

SCHEMBL4667859

CC(C)N(N)C(=O)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 3/20 0.47
HSD11B1 P28845 1/20 0.47
MLYCD O95822 1/20 0.46
ALDH1A1 P00352 4/20 0.43
MAPT P10636 2/20 0.43
TSHR P16473 2/20 0.43
POLB P06746 2/20 0.43
HPGD P15428 1/20 0.43
CYP3A4 P08684 1/20 0.43
PARP1 P09874 1/20 0.43
CYP2C19 P33261 1/20 0.43
RECQL P46063 1/20 0.43
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
PGR P06401 1/20 0.43
ADRA2A P08913 1/20 0.43
ADRA2B P18089 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7371261 0.84 TRPM8 (0.45) TRPM8HSD11B1MLYCDALDH1A1MAPT
SCHEMBL28320439 0.84 TRPM8 (0.45) TRPM8HSD11B1MLYCDALDH1A1MAPT
SCHEMBL10904843 0.82 TRPM8 (0.59) TRPM8ALDH1A1TDP1L3MBTL1LMNA
SCHEMBL28182286 0.82 TRPM8 (0.59) TRPM8ALDH1A1TDP1L3MBTL1LMNA
SCHEMBL28336781 0.82 CA1 (0.46) ALDH1A1MAPTHPGDCYP3A4BLM
SCHEMBL28266347 0.81 TRPM8 (0.43) TRPM8HSD11B1MLYCDALDH1A1MAPT
SCHEMBL9508600 0.81 TRPM8 (0.47) TRPM8ALDH1A1MAPTTSHRHPGD
SCHEMBL19418154 0.80 NPSR1 (0.37) TRPM8MLYCDALDH1A1HPGDL3MBTL1
SCHEMBL4000774 0.80 KDM4E (0.47) MLYCDALDH1A1TSHRHPGDCYP3A4
SCHEMBL18988683 0.80 MLYCD (0.48) TRPM8HSD11B1MLYCDALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107445920-A A kind of production method of bentazone raw pesticide 江苏绿叶农化有限公司 2017-12-08 CN claimed
WO-2023097386-A1 SELECTIVE HDAC6-INHIBITING N-ACYLHYDRAZONE COMPOUNDS, METHODS FOR PRODUCING SAME, COMPOSITIONS, USES, TREATMENT METHODS AND KITS EUROFARMA LABORATÓRIOS S.A (BR) 2023-06-08 WO disclosed
CN-107445920-A A kind of production method of bentazone raw pesticide 江苏绿叶农化有限公司 2017-12-08 CN disclosed
WO-2010115264-A1 INHIBITORS OF HIV REPLICATION BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-10-14 WO disclosed
EP-2004615-A2 QUINAZOLINES FOR PDK1 INHIBITION Novartis AG (CH) 2008-12-24 EP disclosed
WO-2007117607-A9 QUINAZOLINES FOR PDK1 INHIBITION NOVARTIS VACCINES & DIAGNOSTIC (US) 2008-03-06 WO disclosed
WO-2007117607-A2 QUINAZOLINES FOR PDK1 INHIBITION NOVARTIS AG (CH) 2007-10-18 WO disclosed
US-6904423-B1 Method and system for artificial intelligence directed lead discovery through multi-domain clustering BIOREASON, INC. (US) 2005-06-07 US disclosed
US-20040117164-A1 Method and system for artificial intelligence directed lead discovery in high throughput screening data BIOREASON, INC. 2004-06-17 US disclosed
US-6625585-B1 Method and system for artificial intelligence directed lead discovery though multi-domain agglomerative clustering BIOREASON, INC. 2003-09-23 US disclosed
US-5354762-A Insecticides ROHM AND HAAS COMPANY (US) 1994-10-11 US disclosed
EP-0361645-B1 ORGANIC HYDRAZINE DERIVATIVES FOR PHARMACEUTICAL USE ROHM AND HAAS COMPANY (US) 1993-09-29 EP disclosed
EP-0261755-B1 FIVE-MEMBERED HETEROCYCLIC DERIVATIVES OF N'-SUBSTITUTED-N,N'-DIACYLHYDRAZINES ROHM AND HAAS COMPANY (US) 1992-12-16 EP disclosed
US-5117057-A Insecticidal N' substituted-N-N'-disubstituted-hydrazines ROHM AND HAAS COMPANY (US) 1992-05-26 US disclosed
EP-0480661-A1 Insecticidal ferrocenoyl acylhydrazines ROHM AND HAAS COMPANY (US) 1992-04-15 EP disclosed
US-5075471-A Plant destroying insects ROHM AND HAAS COMPANY (US) 1991-12-24 US disclosed
EP-0253468-B1 SIX-MEMBERED HETEROCYCLIC DERIVATIVES OF N'SUBSTITUTED-N,N'-DIACYLHYDRAZINES ROHM AND HAAS COMPANY (US) 1991-11-06 EP disclosed
EP-0361645-A2 Organic hydrazine derivatives for pharmaceutical use ROHM AND HAAS COMPANY (US) 1990-04-04 EP disclosed
EP-0261755-A2 Five-membered heterocyclic derivatives of N'-substituted-N,N'-Diacylhydrazines ROHM AND HAAS COMPANY (US) 1988-03-30 EP disclosed
EP-0253468-A2 Six-membered heterocyclic derivatives of N'substituted-N,N'-diacylhydrazines ROHM AND HAAS COMPANY (US) 1988-01-20 EP disclosed