SCHEMBL4672579

SCHEMBL4672579

O=C(C=C(O)c1nc[nH]n1)c1occ(CCc2ccccc2)c1Cc1ccncc1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.35
GPR52 Q9Y2T5 1/20 0.34
LTA4H P09960 1/20 0.33
DAO P14920 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PLA2G7 Q13093 2/20 0.32
CYP19A1 P11511 2/20 0.32
CYP11B1 P15538 2/20 0.32
CYP11B2 P19099 2/20 0.32
CYP17A1 P05093 1/20 0.32
RAB9A P51151 1/20 0.31
KDM4E B2RXH2 1/20 0.31
HIF1A Q16665 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4671359 0.94 GPR52 (0.35) ABCB1GPR52LTA4HDAOSMN1; SMN2
SCHEMBL4680185 0.90 LMNA (0.35) DAORAB9AKDM4E
SCHEMBL4675251 0.85 ABCB1 (0.35) ABCB1GPR52LTA4HDAOSMN1; SMN2
SCHEMBL4672755 0.84 ALDH1A1 (0.32)
SCHEMBL4673697 0.84 DAO (0.35) GPR52DAORAB9A
SCHEMBL4673674 0.84
SCHEMBL4674138 0.84 LMNA (0.31)
SCHEMBL4673237 0.83 GPR52 (0.34) ABCB1GPR52LTA4HSMN1; SMN2PLA2G7
SCHEMBL5899405 0.83 GPR52 (0.34) ABCB1GPR52LTA4HDAOSMN1; SMN2
SCHEMBL4675675 0.83 LMNA (0.35) DAORAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1142872-B1 AROMATIC HETEROCYCLE COMPOUNDS HAVING HIV INTEGRASE INHIBITING ACTIVITIES SHIONOGI & CO (JP) 2008-10-15 EP disclosed
US-6645956-B1 1-(5-(4-fluorobenzyl)furan-2-yl)-3-hydroxy-3-(1H-1,2,4-triazol-3 -yl)-propenone; viricides; AIDS treatment SHIONOGI & CO., LTD. (JP) 2003-11-11 US disclosed
US-6620841-B1 Furan or benzofuran derivatives substituted with triazole; acquired immunodeficiency syndrome (AIDS) SHIONOGI & CO., LTD. (JP) 2003-09-16 US disclosed
CN-1335834-A Aromatic heterocyclic compounds having HIV integrase inhibitory activity SHIONOGI & CO (JP) 2002-02-13 CN disclosed
EP-1142872-A1 AROMATIC HETEROCYCLE COMPOUNDS HAVING HIV INTEGRASE INHIBITING ACTIVITIES SHIONOGI & CO., LTD. (JP) 2001-10-10 EP disclosed