SCHEMBL4672927

SCHEMBL4672927

CN(C(=O)OC(C)(C)C)C1(CNc2ccc(Cl)nc2)CC1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 1/20 0.36
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
RAB9A P51151 1/20 0.34
GAA P10253 1/20 0.34
LMNA P02545 1/20 0.34
P2RX3 P56373 1/20 0.34
KCNQ3 O43525 7/20 0.34
KCNQ2 O43526 7/20 0.34
KCNE1 P15382 3/20 0.34
KCNQ1 P51787 3/20 0.34
AAK1 Q2M2I8 1/20 0.33
FPR2 P25090 1/20 0.33
BACE1 P56817 1/20 0.33
DRD2 P14416 1/20 0.33
MAPT P10636 1/20 0.33
TSHR P16473 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4793425 0.87 CYP26A1 (0.36) MEN1KMT2AAAK1FPR2MAPT
SCHEMBL4818195 0.83 KCNQ3 (0.41) ALDH1A1MEN1KMT2ARAB9ALMNA
SCHEMBL4669026 0.79 TNF (0.38) ALDH1A1MEN1KMT2ALMNAKCNQ3
Hydrochloric Acid SCHEMBL4823521 0.78 TNF (0.37) ALDH1A1MEN1KMT2ALMNA
SCHEMBL3785603 0.76 FNTA (0.37) P2RX3
SCHEMBL3768495 0.74 SSTR5 (0.37) AAK1
SCHEMBL3776782 0.72 CHEK1 (0.41) AAK1
SCHEMBL3781094 0.70 KMO (0.38) MEN1KMT2ARAB9A
SCHEMBL29819093 0.70 POLB (0.40) ALDH1A1SMN1; SMN2
SCHEMBL4817839 0.70 GRM5 (0.39) ALDH1A1RAB9AGAAKCNQ3KCNQ2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1757586-B1 POLYSBUSTITUIRTE 1,1-PYRIDINYLAMINOCYCLOPROPANAMIN DERIVATE, VERFAHREN ZU DEREN HERSTELLUNG UND DIESE ENTHALTENDE PHARMATUETISCHE ZUSAMMENSETZUNG SERVIER LAB (FR) 2008-12-03 EP disclosed
EP-1757586-A1 POLYSBUSTITUIRTE 1,1-PYRIDINYLAMINOCYCLOPROPANAMIN DERIVATE, VERFAHREN ZU DEREN HERSTELLUNG UND DIESE ENTHALTENDE PHARMATUETISCHE ZUSAMMENSETZUNG Les Laboratoires Servier (FR) 2007-02-28 EP disclosed