SCHEMBL4673017

SCHEMBL4673017

c1ccc(CC2(CNc3cccnc3)CC2)cc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.50
CYP3A4 P08684 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C19 P33261 1/20 0.44
HTR2C P28335 1/20 0.44
RAB9A P51151 3/20 0.43
GRIN2B Q13224 1/20 0.42
BCL6 P41182 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
PKM P14618 3/20 0.40
NPC1 O15118 1/20 0.40
CFTR P13569 1/20 0.40
GOPC Q9HD26 1/20 0.40
HPGD P15428 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4805011 0.74 LTA4H (0.79) LTA4HCYP3A4CYP2D6CYP2C9CYP1A2
SCHEMBL4670579 0.73 BCDIN3D (0.55) LTA4HRAB9APKMNPC1CFTR
SCHEMBL13389708 0.73 HTR2C (0.45) LTA4HCYP3A4CYP2D6CYP2C9CYP1A2
SCHEMBL18458974 0.72 CHRNB2 (0.46) HTR2CSMN1; SMN2
SCHEMBL4670501 0.72 SMN1; SMN2 (0.45) LTA4HCYP3A4CYP2D6CYP2C9RAB9A
Hydrochloric Acid SCHEMBL4826139 0.72 BCDIN3D (0.54) LTA4HRAB9AHPGDMEN1KMT2A
SCHEMBL15904401 0.71 L3MBTL1 (0.63) LTA4HCYP3A4CYP2D6CYP2C9CYP1A2
SCHEMBL8362789 0.71 CHRNB2 (0.47) CYP2D6CYP1A2RAB9APKMMEN1
SCHEMBL4669074 0.71 RAB9A (0.46) LTA4HRAB9ASMN1; SMN2HPGD
SCHEMBL4669084 0.71 RAB9A (0.46) LTA4HRAB9ASMN1; SMN2HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1757586-B1 POLYSBUSTITUIRTE 1,1-PYRIDINYLAMINOCYCLOPROPANAMIN DERIVATE, VERFAHREN ZU DEREN HERSTELLUNG UND DIESE ENTHALTENDE PHARMATUETISCHE ZUSAMMENSETZUNG SERVIER LAB (FR) 2008-12-03 EP disclosed
EP-1757586-A1 POLYSBUSTITUIRTE 1,1-PYRIDINYLAMINOCYCLOPROPANAMIN DERIVATE, VERFAHREN ZU DEREN HERSTELLUNG UND DIESE ENTHALTENDE PHARMATUETISCHE ZUSAMMENSETZUNG Les Laboratoires Servier (FR) 2007-02-28 EP disclosed