Ethylene

Ethylene

SCHEMBL4676980

C=C.CSc1cccc(C23CCC(=O)CC2C3)c1

nearest known ligand 0.42

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.33
CYP2C9 P11712 1/20 0.33
KMT2A Q03164 1/20 0.33
ALDH1A1 P00352 3/20 0.32
CYP3A4 P08684 3/20 0.32
MAPT P10636 1/20 0.32
CFTR P13569 1/20 0.31
SIGMAR1 Q99720 2/20 0.31
MGLL Q99685 1/20 0.31
THRB P10828 1/20 0.30
MAPK1 P28482 1/20 0.30
DDB1 Q16531 1/20 0.30
CRBN Q96SW2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4679336 0.97 MEN1 (0.35) MEN1CYP2C9KMT2AALDH1A1CYP3A4
Ethylene SCHEMBL4673356 0.79 ALDH1A1 (0.32) ALDH1A1CYP3A4MAPTSIGMAR1MGLL
Ethylene SCHEMBL4679206 0.77 MCHR1 (0.39) DDB1CRBN
SCHEMBL25635537 0.77 KDM1A (0.44) MEN1CYP2C9KMT2ACYP3A4
SCHEMBL14336703 0.76 MEN1 (0.48) MEN1CYP2C9KMT2AALDH1A1CYP3A4
Ethylene SCHEMBL4679116 0.74 MEN1 (0.41) MEN1CYP2C9KMT2AALDH1A1MAPT
SCHEMBL4674917 0.74 HSD11B1 (0.41) DDB1CRBN
SCHEMBL14102149 0.72 OPRD1 (0.32)
Ethylene SCHEMBL4674837 0.71 HPGDS (0.35) MGLL
SCHEMBL614812 0.71 MEN1 (0.43) MEN1CYP2C9KMT2AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1453501-B1 N- ARYL-N'-ARYLCYCLOALKYL-UREA DERIVATIVES AS MCH ANTAGONISTS FOR THE TREATMENT OF OBESITY SCHERING CORP (US) 2008-08-13 EP disclosed
US-7348328-B2 MCH antagonists for the treatment of obesity SCHERING CORPORATION (US) 2008-03-25 US disclosed
EP-1453501-A1 N- ARYL-N'-ARYLCYCLOALKYL-UREA DERIVATIVES AS MCH ANTAGONISTS FOR THE TREATMENT OF OBESITY SCHERING CORPORATION (US) 2004-09-08 EP disclosed
US-20040122017-A1 MCH antagonists for the treatment of obesity SCHERING CORPORATION 2004-06-24 US disclosed
WO-2003047568-A1 N-ARYL-N'-ARYLCYCLOALKYL-UREA DERIVATIVES AS MCH ANTAGONISTS FOR THE TREATMENT OF OBESITY SCHERING CORPORATION (US) 2003-06-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040122017-A1 MCH antagonists for the treatment of obesity MCHR1, MCHR2, MC4R MEN1 457/4885CYP2C9 3104/4885KMT2A 225/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.