SCHEMBL4677322

SCHEMBL4677322

O=C(O)C(C(=O)O)C1CN(C(c2ccccc2)c2ccccc2)C1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
KMT2A Q03164 3/20 0.47
SLC6A9 P48067 1/20 0.47
MAOB P27338 1/20 0.46
CYP3A4 P08684 2/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
KDM4E B2RXH2 2/20 0.45
MAPT P10636 2/20 0.45
HPGD P15428 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
CNR1 P21554 1/20 0.44
CNR2 P34972 1/20 0.44
CACNA2D1 P54289 2/20 0.44
CACNA1B Q00975 2/20 0.44
CACNB1 Q02641 2/20 0.44
CACNA1C Q13936 2/20 0.44
MEN1 O00255 1/20 0.44
CACNA1H O95180 1/20 0.44
OPRD1 P41143 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11455106 0.84 ALDH1A1 (0.46) ALDH1A1KMT2ASLC6A9MAOBKDM4E
SCHEMBL1661498 0.80 CACNA2D1 (0.51) KMT2ASLC6A9KDM4ENPSR1CACNA2D1
SCHEMBL3421906 0.80 MAPT (0.41) ALDH1A1KMT2ASLC6A9CYP3A4CYP2D6
SCHEMBL85386 0.78 ALDH1A1 (0.54) ALDH1A1KMT2ASLC6A9MAOBKDM4E
SCHEMBL20594076 0.76 KMT2A (0.57) ALDH1A1KMT2ASLC6A9MAOBCYP3A4
SCHEMBL29220868 0.76 SLC6A9 (0.44) ALDH1A1KMT2ASLC6A9MAOBCYP2D6
SCHEMBL5074961 0.76 KMT2A (0.45) ALDH1A1KMT2ASLC6A9MAOBMAPT
SCHEMBL4321754 0.76 OPRM1 (0.51) ALDH1A1KMT2ASLC6A9MAOBCYP3A4
SCHEMBL16448458 0.76 OPRM1 (0.50) ALDH1A1KMT2ASLC6A9CYP2D6NPSR1
SCHEMBL12499368 0.75 ALDH1A1 (0.51) ALDH1A1KMT2ASLC6A9MAOBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1304329-B1 Pyridonecarboxylic acid derivatives and their use as antibacterial agents DAIICHI SANKYO CO LTD (JP) 2008-10-15 EP disclosed
EP-1304329-A2 Pyridonecarboxylic acid derivatives and their use as antibacterial agents DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2003-04-23 EP disclosed
US-5849757-A Pyridonecarboxylic acid derivatives substituted by a bicyclic amino group as antibacterials DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1998-12-15 US disclosed
EP-0807630-A1 HETEROCYCLIC COMPOUNDS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1997-11-19 EP disclosed