SCHEMBL4680128

SCHEMBL4680128

N#Cc1ccc(CO)c(C(=O)O)c1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 1/20 0.44
XDH P47989 2/20 0.43
SLC22A12 Q96S37 2/20 0.43
HTT P42858 2/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.40
MAP2K1 Q02750 1/20 0.40
PIN1 Q13526 1/20 0.40
NOTUM Q6P988 1/20 0.39
ALB P02768 1/20 0.39
FFAR1 O14842 1/20 0.38
TRPM4 Q8TD43 1/20 0.38
HNF4A P41235 1/20 0.38
MCL1 Q07820 1/20 0.37
GSK3B P49841 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23480907 0.86 SLC22A12 (0.46) CDK2XDHSLC22A12HTTPTGDR2
SCHEMBL18398646 0.84 GSK3B (0.43) CDK2XDHSLC22A12HTTPTGDR2
SCHEMBL13291209 0.80 ALB (0.41) CDK2XDHSLC22A12HTTMAP2K1
SCHEMBL27752918 0.79 GABRP (0.44) CDK2XDHSLC22A12NOTUMFFAR1
SCHEMBL3157619 0.79 XDH (0.53) XDHSLC22A12HTTMAP2K1PIN1
SCHEMBL13608787 0.77 CA2 (0.41) PTGDR2NOTUM
SCHEMBL7196160 0.76 XDH (0.46) XDHSLC22A12HTTMAP2K1PIN1
SCHEMBL30902488 0.76 HNF4A (0.62) XDHSLC22A12HTTHNF4AMCL1
SCHEMBL131551 0.76 HNF4A (0.62) XDHSLC22A12HTTHNF4AMCL1
SCHEMBL1232210 0.76 MEN1 (0.47) HTTPTGDR2ALBGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102596921-B Novel compounds GLAXO GROUP LTD 2015-04-29 CN disclosed
CN-104292154-A Novel compounds GLAXO GROUP LTD 2015-01-21 CN disclosed
CN-103221047-B Compounds and methods TEMPERO PHARMACEUTICALS INC 2014-12-17 CN disclosed
CN-101970420-B Oxadiazole derivatives MERCK SERONO SA 2014-09-24 CN disclosed
CN-102272111-A 1,2 -thiazol yl derivatives as cannabinoid receptor ligands 2011-12-07 CN disclosed
CN-101970420-A Oxadiazole derivatives MERCK SERONO SA 2011-02-09 CN disclosed
CN-101765594-A 1,3-thiazoles-2 (3H)-ylidene compounds as cannabinoid receptor ligand ABBOTT LAB 2010-06-30 CN disclosed
CN-101765593-A 2-iminoisothiazole derivatives as cannabinoid receptor ligands ABBOTT LAB 2010-06-30 CN disclosed
EP-1362856-B1 WATER-SOLUBLE TRIAZOLE FUNGICIDE DAIICHI SANKYO CO LTD (JP) 2008-09-10 EP disclosed
CN-1144805-C Bispidine compounds useful in treatment of cardiac arrhythmias 2004-04-07 CN disclosed
CN-1284956-A Novel bispidine antiarrhythmic compounds ASTRA ZENECA AKTIEBOLAG (SE) 2001-02-21 CN disclosed