SCHEMBL4680942

SCHEMBL4680942

CS(=O)(=O)OC(Br)c1c(F)cccc1F

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
ALDH1A1 P00352 2/20 0.32
PKM P14618 1/20 0.32
PKLR P30613 1/20 0.32
GRIA4 P48058 1/20 0.31
HTT P42858 1/20 0.31
LMNA P02545 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.30
PSIP1 O75475 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1604902 0.79 ALDH1A1 (0.38) CES2CES1ALDH1A1PKMPKLR
SCHEMBL17185881 0.74 ALDH1A1 (0.33) CES2CES1ALDH1A1PKMPKLR
SCHEMBL19717529 0.74 CES2 (0.39) CES2CES1ALDH1A1HTT
SCHEMBL7957999 0.71 CES2 (0.39) CES2CES1ALDH1A1LMNA
SCHEMBL6258207 0.67 MC4R (0.40) CES2CES1ALDH1A1SMN1; SMN2
SCHEMBL4828643 0.66 CES2 (0.39) CES2CES1
SCHEMBL18242776 0.66 CES2 (0.43) CES2CES1ALDH1A1LMNASMN1; SMN2
SCHEMBL6204096 0.66 CES2 (0.39) CES2CES1ALDH1A1SMN1; SMN2
SCHEMBL3755699 0.66 PKM (0.36) CES2CES1ALDH1A1PKMPKLR
Methanesulfonic Acid Methyl Ester SCHEMBL27591830 0.66 USP2 (0.46) CES2CES1ALDH1A1PKMPKLR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1915373-A1 HETEROBICYCLIC COMPOUNDS USEFUL AS P38 KINASE INHIBITING AGENTS Merck and Co., Inc. (US) 2008-04-30 EP disclosed
WO-2007021710-A1 HETEROBICYCLIC COMPOUNDS USEFUL AS P38 KINASE INHIBITING AGENTS MERCK & CO., INC. (US) 2007-02-22 WO disclosed