SCHEMBL4681340

SCHEMBL4681340

CS(=O)(=O)N(CCN)c1ccccc1N1CCN(C(=O)[C@@H](Cc2ccc(Cl)cc2)N2[CH]Cc3ccccc3C2)CC1

nearest known ligand 0.51

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
MC4R P32245 20/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4684460 0.90 MC4R (0.55) MC4R
SCHEMBL5478550 0.83 MC4R (0.59) MC4R
SCHEMBL4681085 0.81 LMNA (0.47) MC4R
SCHEMBL4681379 0.80 MC4R (0.49) MC4R
SCHEMBL4681339 0.80 MC4R (0.47) MC4R
SCHEMBL4784715 0.78 MC4R (0.45) MC4R
SCHEMBL4685109 0.77 MC4R (0.42) MC4R
SCHEMBL4514886 0.75 MC4R (0.67) MC4R
SCHEMBL4514892 0.75 MC4R (0.60) MC4R
SCHEMBL4531987 0.74 TACR1 (0.56) MC4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1417190-B1 SUBSTITUTED PIPERAZINES AS MODULATORS OF THE MELANOCORTIN RECEPTOR AMGEN INC (US) 2008-10-22 EP disclosed