SCHEMBL4684141

SCHEMBL4684141

Cc1cc(S(=O)(=O)OCCO)cc(C)c1C

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.37
GAA P10253 2/20 0.31
PDK1 Q15118 1/20 0.31
PDK2 Q15119 1/20 0.31
PDK3 Q15120 1/20 0.31
PDK4 Q16654 1/20 0.31
HTT P42858 3/20 0.31
STAT3 P40763 1/20 0.31
FABP4 P15090 1/20 0.30
PDIA6 Q15084 1/20 0.30
LMNA P02545 1/20 0.30
MAPK1 P28482 1/20 0.30
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8923981 0.85 ALDH1A1 (0.36) ALDH1A1GAAHTTSTAT3FABP4
SCHEMBL4684137 0.83 KDM4E (0.32) ALDH1A1HTTPDIA6LMNACA12
SCHEMBL8923591 0.82 LMNA (0.47) ALDH1A1GAAHTTLMNA
SCHEMBL8923976 0.79 LMNA (0.32) ALDH1A1GAALMNAMAPK1
SCHEMBL4686793 0.77 TSHR (0.33) ALDH1A1LMNAMAPK1
SCHEMBL1258986 0.76 STAT3 (0.47) ALDH1A1GAASTAT3CA12CA1
Dimethylamine SCHEMBL28544509 0.75 STAT3 (0.47) ALDH1A1GAAHTTSTAT3LMNA
SCHEMBL1832458 0.74 KMT2A (0.47) ALDH1A1GAA
Ethylene SCHEMBL7519766 0.73 STAT3 (0.44) ALDH1A1GAASTAT3CA12CA1
Ethylene SCHEMBL11280661 0.73 STAT3 (0.44) ALDH1A1GAASTAT3CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902717-A2 Vasopressin antagonist and oxytocin antagonist Otsuka Pharmaceutical Company, Limited (JP) 2008-03-26 EP disclosed
EP-0620003-B1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMA CO LTD (JP) 2008-01-16 EP disclosed
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5622947-A VASODILATORS, HYPOTENSIVE AGENTS, DIURETICS, PLATELET AGGLUTINATION INHIBITORS; ALSO USED TO PREVENT PREMATURE BIRTH, TREAT DYSMENORRHEA OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-04-22 US disclosed
EP-0514667-B1 Benzazepin derivatives as vasopressin antagonists OTSUKA PHARMA CO LTD (JP) 1995-08-09 EP disclosed
EP-0620003-A1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed
US-5244898-A Vasopressin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1993-09-14 US disclosed
EP-0514667-A1 Benzazepin derivatives as vasopressin antagonists OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-11-25 EP disclosed