SCHEMBL4684155

SCHEMBL4684155

CCOc1ccc(CCCC(N)=O)cc1OCC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
GAA P10253 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.49
KMT2A Q03164 2/20 0.49
MEN1 O00255 1/20 0.48
MAPK1 P28482 1/20 0.48
CYP2C19 P33261 3/20 0.47
CYP2C9 P11712 2/20 0.47
CYP3A4 P08684 1/20 0.47
POLB P06746 1/20 0.47
CYP1A2 P05177 1/20 0.47
MAPT P10636 1/20 0.47
CALM1 P0DP23 2/20 0.47
BIRC5 O15392 1/20 0.47
LMNA P02545 1/20 0.46
CYP2D6 P10635 1/20 0.46
F2 P00734 1/20 0.46
F10 P00742 1/20 0.46
PRSS1 P07477 1/20 0.46
F7 P08709 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30303113 0.88 PPARG (0.52) MAPK1CYP2C19CYP2C9CYP3A4CYP1A2
SCHEMBL5723918 0.88 CYP1A2 (0.48) ALDH1A1GAAKMT2AMEN1MAPK1
SCHEMBL8501979 0.86 MAPK1 (0.54) KMT2AMEN1MAPK1CALM1
SCHEMBL4684153 0.86 GAA (0.49) ALDH1A1GAAKMT2AMEN1CYP2C19
SCHEMBL28323456 0.84 L3MBTL1 (0.54) KMT2AMEN1CALM1
SCHEMBL27773869 0.83 PPARA (0.50) ALDH1A1GAAKMT2AMEN1CYP2C19
SCHEMBL11911909 0.83 BIRC5 (0.62) ALDH1A1GAASMN1; SMN2KMT2AMEN1
SCHEMBL30303108 0.82 CYP1A2 (0.52) ALDH1A1CYP2C19CYP2C9CYP3A4CYP1A2
SCHEMBL2224074 0.82 ATM (0.61) ALDH1A1KMT2APOLB
SCHEMBL29463761 0.82 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2KMT2AMAPK1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902717-A2 Vasopressin antagonist and oxytocin antagonist Otsuka Pharmaceutical Company, Limited (JP) 2008-03-26 EP disclosed
EP-0620003-B1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMA CO LTD (JP) 2008-01-16 EP disclosed
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5622947-A VASODILATORS, HYPOTENSIVE AGENTS, DIURETICS, PLATELET AGGLUTINATION INHIBITORS; ALSO USED TO PREVENT PREMATURE BIRTH, TREAT DYSMENORRHEA OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-04-22 US disclosed
EP-0514667-B1 Benzazepin derivatives as vasopressin antagonists OTSUKA PHARMA CO LTD (JP) 1995-08-09 EP disclosed
EP-0620003-A1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed
US-5244898-A Vasopressin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1993-09-14 US disclosed
EP-0514667-A1 Benzazepin derivatives as vasopressin antagonists OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-11-25 EP disclosed