SCHEMBL5723918

SCHEMBL5723918

CCOc1cc(CCCC(N)=O)ccc1O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2C8 P10632 2/20 0.48
CYP2C9 P11712 2/20 0.48
CYP2B6 P20813 2/20 0.48
CYP2C19 P33261 2/20 0.48
ALOX5 P09917 3/20 0.48
OR51E2 Q9H255 1/20 0.48
ALDH1A1 P00352 3/20 0.48
MTNR1A P48039 1/20 0.47
MTNR1B P49286 1/20 0.47
TSHR P16473 3/20 0.46
TAAR1 Q96RJ0 2/20 0.46
MAPK1 P28482 1/20 0.46
KDM4E B2RXH2 2/20 0.46
TOP2A P11388 1/20 0.46
LMNA P02545 1/20 0.45
GLA P06280 1/20 0.45
HTR1A P08908 3/20 0.44
TRPV1 Q8NER1 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30303108 0.94 CYP1A2 (0.52) CYP1A2CYP3A4CYP2C8CYP2C9CYP2B6
SCHEMBL4684155 0.88 ALDH1A1 (0.50) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL5723843 0.85 ALOX5 (0.66) CYP1A2CYP3A4CYP2C8CYP2C9CYP2B6
SCHEMBL20399514 0.83 ALDH1A1 (0.51) CYP1A2CYP3A4CYP2C8CYP2C9CYP2B6
SCHEMBL29610155 0.82 ALOX5 (0.54) CYP1A2CYP3A4CYP2C8CYP2C9CYP2B6
SCHEMBL12799076 0.82 ALOX5 (0.54) CYP1A2CYP3A4CYP2C8CYP2C9CYP2B6
SCHEMBL6583668 0.82 ALOX5 (0.54) CYP1A2CYP3A4CYP2C8CYP2C9CYP2B6
SCHEMBL8890692 0.82 ALOX5 (0.49) CYP1A2CYP3A4CYP2C8CYP2C9CYP2B6
SCHEMBL20399450 0.81 KAT8 (0.53) CYP1A2CYP3A4CYP2C8CYP2C9CYP2B6
SCHEMBL12788915 0.81 TSHR (0.69) CYP1A2CYP3A4ALDH1A1MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633715-A1 2-(6-AMINO-PYRIDIN-3-YL)-2-HYDROXYETHYLAMINE DERIVATIVES AS BETA 2-ADRENOCEPTORS AGONISTS Pfizer Limited (GB) 2006-03-15 EP disclosed
WO-2004108676-A1 2-(6-AMINO-PYRIDIN-3-YL)-2-HYDROXYETHYLAMINE DERIVATIVES AS BETA 2-ADRENOCEPTORS AGONISTS PFIZER LIMITED (GB) 2004-12-16 WO disclosed