SCHEMBL4685647

SCHEMBL4685647

CCC1(O)CCCCC1(OC(F)(F)F)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33
PRCP P42785 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
ALDH1A1 P00352 2/20 0.33
TACR1 P25103 1/20 0.33
POLB P06746 1/20 0.33
SLC6A4 P31645 2/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A3 Q01959 1/20 0.33
DPP4 P27487 1/20 0.33
AKR1C1 Q04828 1/20 0.33
APOBEC3A P31941 2/20 0.32
APOBEC3G Q9HC16 2/20 0.32
HTT P42858 1/20 0.32
CCR6 P51684 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM1 P11229 1/20 0.32
DRD3 P35462 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4984844 0.82 SLC6A4 (0.38) OPRM1PRCPSIGMAR1ALDH1A1POLB
SCHEMBL6470519 0.78 TACR1 (0.35) OPRM1OPRD1OPRK1PRCPSIGMAR1
SCHEMBL4540372 0.77 OPRL1 (0.39) OPRM1OPRD1OPRK1TACR1SLC6A4
SCHEMBL4991848 0.76 TRPA1 (0.36) OPRM1SLC6A4SLC6A2SLC6A3DPP4
SCHEMBL5695494 0.69 OPRM1 (0.36) OPRM1OPRD1OPRK1POLB
SCHEMBL10618939 0.67 SLC6A4 (0.50) OPRM1OPRK1SLC6A4SLC6A2SLC6A3
SCHEMBL3521192 0.64 SLC6A4 (0.44) POLBSLC6A4SLC6A2SLC6A3CCR6
SCHEMBL4636975 0.63 AKR1C1 (0.35) OPRM1OPRD1OPRK1AKR1C1HTT
SCHEMBL5538611 0.62 AKR1C1 (0.38) OPRM1PRCPSIGMAR1ALDH1A1POLB
SCHEMBL4543656 0.62 TACR1 (0.39) OPRM1OPRD1OPRK1TACR1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957470-A1 PROCESS FOR SELECTIVE SYNTHESIS OF ENANTIOMERS OF SUBSTITUTED 1-(2-AMINO-1-PHENYL-ETHYL)-CYCLOHEXANOLS Wyeth (US) 2008-08-20 EP disclosed
WO-2007067501-A1 PROCESS FOR SELECTIVE SYNTHESIS OF ENANTIOMERS OF SUBSTITUTED 1-(2-AMINO-1-PHENYL-ETHYL)-CYCLOHEXANOLS WYETH (US) 2007-06-14 WO disclosed
EP-1673059-A2 ALKANOL AND CYCLOALKANOL-AMINE DERIVATIVES AND METHODS OF THEIR USE Wyeth (US) 2006-06-28 EP disclosed
EP-1673090-A1 FUSED-ARYL AND HETEROARYL DERIVATIVES AND METHODS OF THEIR USE Wyeth (US) 2006-06-28 EP disclosed
WO-2005037207-A2 ARYLALKYL-PIPERAZINE DERIVATIVES FOR THE TREATMENT OF CONDITIONS AMELIORATED BY MONOAMINE REUPTAKE INCLUDING VASOMOTOR SYMPTOMS (VMS) WYETH (US) 2005-04-28 WO disclosed
WO-2005037283-A1 FUSED-ARYL AND HETEROARYL DERIVATIVES AND METHODS OF THEIR USE WYETH (US) 2005-04-28 WO disclosed