SCHEMBL4687910

SCHEMBL4687910

NC(=O)CCOc1ccccn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.46
LTB4R Q15722 1/20 0.43
NPC1 O15118 2/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
GRM2 Q14416 1/20 0.40
PARP10 Q53GL7 1/20 0.40
PSMB5 P28074 1/20 0.39
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
DRD3 P35462 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
PDK2 Q15119 1/20 0.38
FURIN P09958 1/20 0.38
LMNA P02545 2/20 0.38
SCN7A Q01118 1/20 0.38
KCNH2 Q12809 1/20 0.38
NAPRT Q6XQN6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5517724 0.84 LMNA (0.50) TSHRLTB4RNPC1RAB9ASMN1; SMN2
SCHEMBL1178753 0.81 TSHR (0.51) TSHRNPC1RAB9ASMN1; SMN2PARP10
SCHEMBL3829038 0.81 LMNA (0.49) TSHRNPC1RAB9ASMN1; SMN2GRM2
SCHEMBL5515476 0.79 LTB4R (0.54) LTB4RSMN1; SMN2ALDH1A1
SCHEMBL31482995 0.78 TSHR (0.43) TSHRNPC1RAB9ASMN1; SMN2PSMB5
SCHEMBL4190714 0.78 KDM4E (0.50) TSHRNPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL5522710 0.77 LTB4R (0.55) LTB4RSMN1; SMN2ALDH1A1
SCHEMBL1178754 0.75 KDM4E (0.50) NPC1RAB9ASMN1; SMN2ALDH1A1CYP2D6
SCHEMBL2416582 0.75 ALDH1A1 (0.50) TSHRNPC1RAB9ASMN1; SMN2GRM2
SCHEMBL15617823 0.75 NPC1 (0.43) TSHRNPC1RAB9ASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1496838-A4 SUBSTITUTED AMIDES MERCK & CO INC (US) 2008-07-02 EP claimed
EP-1496838-A2 SUBSTITUTED AMIDES Merck & Co., Inc. (US) 2005-01-19 EP claimed
WO-2003077847-A2 SUBSTITUTED AMIDES MERCK & CO., INC. (US) 2003-09-25 WO claimed
EP-1496838-A4 SUBSTITUTED AMIDES MERCK & CO INC (US) 2008-07-02 EP disclosed
EP-1496838-A2 SUBSTITUTED AMIDES Merck & Co., Inc. (US) 2005-01-19 EP disclosed
WO-2003077847-A2 SUBSTITUTED AMIDES MERCK & CO., INC. (US) 2003-09-25 WO disclosed