SCHEMBL4689271

SCHEMBL4689271

CC(c1ccc(Cl)cc1)C(CNC(=O)CC1CC1)c1ccc(Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.48
NPC1 O15118 4/20 0.48
IDO1 P14902 1/20 0.44
HPGD P15428 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
GAA P10253 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TRPV1 Q8NER1 1/20 0.39
KCNH2 Q12809 2/20 0.39
MCHR1 Q99705 1/20 0.39
FFAR2 O15552 1/20 0.38
FDFT1 P37268 1/20 0.38
PRCP P42785 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
OPRM1 P35372 1/20 0.37
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
ALOX12 P18054 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694021 0.78 RAB9A (0.43) RAB9ANPC1SMN1; SMN2MEN1KMT2A
SCHEMBL5266049 0.77 RAB9A (0.60) RAB9ANPC1HPGDSMN1; SMN2MEN1
SCHEMBL13113988 0.76 RAB9A (0.54) RAB9ANPC1IDO1SMN1; SMN2KCNH2
SCHEMBL13804814 0.75 FDFT1 (0.62) RAB9ANPC1FDFT1
SCHEMBL3525023 0.75 FDFT1 (0.62) RAB9ANPC1FDFT1
SCHEMBL4694805 0.74 KMT2A (0.44) RAB9AHPGDSMN1; SMN2MEN1KMT2A
SCHEMBL5201159 0.74 PKM (0.48) RAB9ANPC1HPGDSMN1; SMN2GAA
SCHEMBL5200358 0.74 SMN1; SMN2 (0.41) RAB9ANPC1HPGDSMN1; SMN2GAA
SCHEMBL4688373 0.74 HSD17B10 (0.46) GAAKCNH2ALDH1A1
SCHEMBL5262774 0.74 SLC6A9 (0.54) RAB9ANPC1SMN1; SMN2GAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1496838-A4 SUBSTITUTED AMIDES MERCK & CO INC (US) 2008-07-02 EP claimed
EP-1496838-A2 SUBSTITUTED AMIDES Merck & Co., Inc. (US) 2005-01-19 EP claimed
WO-2003077847-A2 SUBSTITUTED AMIDES MERCK & CO., INC. (US) 2003-09-25 WO claimed