SCHEMBL4689907

SCHEMBL4689907

O=C(O)Oc1ccc2c(c1)N(c1cc(Cl)cc(Cl)c1)C(=O)C2Cc1ccc(Br)cc1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGAL P20701 14/20 0.36
ITGB2 P05107 13/20 0.36
ICAM1 P05362 13/20 0.36
POLB P06746 1/20 0.35
ALOX5 P09917 1/20 0.35
PPARG P37231 1/20 0.34
PPARA Q07869 1/20 0.34
CES2 O00748 1/20 0.34
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692140 0.84 ITGAL (0.38) ITGALITGB2ICAM1ALOX5CES2
SCHEMBL4692248 0.79 ALOX5 (0.47) ITGALITGB2ICAM1ALOX5CES2
SCHEMBL4690047 0.73 ITGAL (0.40) ITGALITGB2ICAM1ALOX5CES2
SCHEMBL4687837 0.73 ITGAL (0.40) ITGALITGB2ICAM1ALOX5CES2
SCHEMBL4687956 0.72 ALOX5 (0.50) ITGALITGB2ICAM1ALOX5CES2
SCHEMBL4690051 0.70 ALOX5 (0.46) ITGALITGB2ICAM1ALOX5CES2
SCHEMBL4693030 0.68 GAA (0.39) ITGALITGB2ICAM1ALOX5CES2
SCHEMBL4687618 0.65 ITGB2 (0.41) ITGALITGB2ICAM1ALOX5CES2
SCHEMBL22898546 0.64 RAB9A (0.58) ITGALITGB2ICAM1
SCHEMBL4689811 0.63 ALOX5 (0.46) ITGALITGB2ICAM1POLBALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1399155-B1 SMALL MOLECULES USEFUL IN THE TREATMENT OF INFLAMMATORY DISEASE BOEHRINGER INGELHEIM PHARMA (US) 2008-05-28 EP claimed