SCHEMBL4690126

SCHEMBL4690126

Cc1ccc(C(CC(N)=O)N2CC3CN(C(=O)c4c(C)n[nH]c4C)CC3C2)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 3/20 0.38
HCRTR2 O43614 3/20 0.38
MAPT P10636 1/20 0.36
EPHX2 P34913 1/20 0.35
FPR2 P25090 6/20 0.35
PROKR1 Q8TCW9 6/20 0.35
TNF P01375 1/20 0.34
NAMPT P43490 2/20 0.34
CCR5 P51681 2/20 0.33
TLR9 Q9NR96 1/20 0.33
TLR8 Q9NR97 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
HRH4 Q9H3N8 1/20 0.33
CCL5 P13501 1/20 0.32
CNR1 P21554 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3283594 0.86 CCL5 (0.43) CCR5CCL5
SCHEMBL3281863 0.85 HCRTR1 (0.48) HCRTR1HCRTR2TNFCCR5
SCHEMBL4690403 0.85 HCRTR1 (0.39) HCRTR1HCRTR2TNFCCR5HRH4
SCHEMBL4694334 0.85 HCRTR1 (0.43) HCRTR1HCRTR2EPHX2TNFCCR5
SCHEMBL4695961 0.85 HCRTR1 (0.36) HCRTR1HCRTR2MAPTTNFCCR5
SCHEMBL3282223 0.85 CCR5 (0.43) HCRTR1HCRTR2CCR5CCL5
SCHEMBL4694265 0.84 HCRTR1 (0.38) HCRTR1HCRTR2FPR2PROKR1TNF
SCHEMBL5659102 0.84 CCR5 (0.45) HCRTR1HCRTR2TNFCCR5HRH4
SCHEMBL4691534 0.84 GFER (0.43) HCRTR1HCRTR2CCR5
SCHEMBL4693896 0.83 HCRTR1 (0.47) HCRTR1HCRTR2MAPTTNFCCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed