SCHEMBL4694265

SCHEMBL4694265

Cc1ccc(C(CC(N)=O)N2CC3CN(C(=O)c4c(C)nn(C)c4C)CC3C2)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 3/20 0.38
HCRTR2 O43614 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
CCR5 P51681 3/20 0.35
POLB P06746 2/20 0.35
TNF P01375 1/20 0.34
FPR2 P25090 1/20 0.34
PROKR1 Q8TCW9 1/20 0.34
NAMPT P43490 2/20 0.34
USP2 O75604 1/20 0.34
LMNA P02545 1/20 0.34
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.34
TLR9 Q9NR96 1/20 0.33
TLR8 Q9NR97 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
CCL5 P13501 4/20 0.33
FNTA P49354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4695130 0.87 KMT2A (0.43) HCRTR1HCRTR2CCR5POLBUSP2
SCHEMBL3283594 0.86 CCL5 (0.43) CCR5CCL5
SCHEMBL3281863 0.85 HCRTR1 (0.48) HCRTR1HCRTR2CCR5TNF
SCHEMBL4690403 0.85 HCRTR1 (0.39) HCRTR1HCRTR2CCR5TNF
SCHEMBL4694334 0.85 HCRTR1 (0.43) HCRTR1HCRTR2CCR5TNFCCL5
SCHEMBL3282223 0.85 CCR5 (0.43) HCRTR1HCRTR2CCR5CCL5
SCHEMBL4694305 0.84 FPR2 (0.50) SMN1; SMN2FPR2PROKR1USP2LMNA
SCHEMBL4690126 0.84 HCRTR1 (0.38) HCRTR1HCRTR2CCR5TNFFPR2
SCHEMBL4691534 0.84 GFER (0.43) HCRTR1HCRTR2SMN1; SMN2NPC1CCR5
SCHEMBL4693079 0.83 HCRTR1 (0.38) HCRTR1HCRTR2CCR5TNFCCL5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed