SCHEMBL4695901

SCHEMBL4695901

COc1ccc(C(=O)N2CC3CN(C(CC(N)=O)c4ccc(C)c(Cl)c4)CC3C2)c(OC)c1

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 16/20 0.47
HCRTR1 O43613 13/20 0.47
HTT P42858 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691836 0.93 HCRTR2 (0.40) HCRTR2HCRTR1HTT
SCHEMBL4690927 0.93 HCRTR1 (0.49) HCRTR2HCRTR1
SCHEMBL4691405 0.90 HCRTR1 (0.48) HCRTR2HCRTR1HTTTSHR
SCHEMBL4690309 0.90 HCRTR1 (0.38) HCRTR2HCRTR1
SCHEMBL4689519 0.88 ALDH1A1 (0.47) HCRTR2HCRTR1
SCHEMBL4693952 0.87 HCRTR1 (0.50) HCRTR2HCRTR1TSHR
SCHEMBL4694424 0.86 HCRTR1 (0.37) HCRTR2HCRTR1
SCHEMBL4692329 0.86 CCR5 (0.44) HCRTR2HCRTR1
SCHEMBL4694350 0.85 KCNK3 (0.42) HCRTR2HCRTR1HTT
SCHEMBL4692627 0.85 HCRTR1 (0.50) HCRTR2HCRTR1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP disclosed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO disclosed