SCHEMBL4690489

SCHEMBL4690489

NC(=O)n1ncc(Cl)c1C(=O)N1CC2CN(CC[CH]c3ccccc3)C[C@H]2C1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.38
KMT2A Q03164 1/20 0.38
CCR5 P51681 14/20 0.36
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA7 P36544 1/20 0.34
CHRNA4 P43681 1/20 0.34
CCL5 P13501 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694169 0.87 PKM (0.37) PKMKMT2ACCR5CHRNB2CHRNB4
SCHEMBL4696786 0.77 CCR5 (0.43) CCR5CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL4694094 0.77 CHRNB2 (0.44) CCR5CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL4693316 0.76 EIF4A3 (0.39) CHRNB2CHRNA7CHRNA4
SCHEMBL4690783 0.76 CCR5 (0.47) CCR5CCL5
SCHEMBL4690864 0.76 RIPK2 (0.40) KMT2A
SCHEMBL4694116 0.76 HCRTR2 (0.38) CCR5CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL4692838 0.75 CCR5 (0.42) CCR5CCL5
SCHEMBL4690459 0.75 MEN1 (0.37) KMT2ACCR5CCL5
SCHEMBL4692781 0.75 PKM (0.36) PKMKMT2ACCR5CHRNB2CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed