SCHEMBL4690459

SCHEMBL4690459

CCc1cc(C(=O)N2CC3CN(CC[CH]c4ccccc4)C[C@H]3C2)n(C(N)=O)n1

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
HCRTR1 O43613 2/20 0.36
HCRTR2 O43614 2/20 0.36
CCL5 P13501 10/20 0.34
CCR5 P51681 6/20 0.33
ALDH1A1 P00352 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4690538 0.80 CCL5 (0.36) HCRTR1HCRTR2CCL5CCR5
SCHEMBL4692820 0.79 CCL5 (0.35) HCRTR1HCRTR2CCL5CCR5ALDH1A1
SCHEMBL4694116 0.76 HCRTR2 (0.38) HCRTR1HCRTR2CCR5
SCHEMBL4691519 0.76 PLA2G10 (0.34) MEN1KMT2AHCRTR1HCRTR2CCR5
SCHEMBL4690155 0.75 MEN1 (0.38) MEN1KMT2ACCL5CCR5ALDH1A1
SCHEMBL4694094 0.75 CHRNB2 (0.44) CCR5ALDH1A1
SCHEMBL4690489 0.75 PKM (0.38) KMT2ACCL5CCR5
SCHEMBL4694287 0.75 CCR5 (0.37) CCL5CCR5
SCHEMBL4693281 0.74 CHRNB2 (0.43) MEN1KMT2ACCR5
SCHEMBL4692781 0.73 PKM (0.36) MEN1KMT2ACCL5CCR5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed