SCHEMBL4690515

SCHEMBL4690515

N#Cc1ccc(C(=O)N2CC3CN(CC[C@H](N)c4ccccc4)CC3C2)cc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
KCNA5 P22460 1/20 0.45
CCR5 P51681 13/20 0.44
CCL5 P13501 3/20 0.43
CCR2 P41597 1/20 0.42
PRKAB2 O43741 1/20 0.40
PRKAG1 P54619 1/20 0.40
PRKAA2 P54646 1/20 0.40
PRKAA1 Q13131 1/20 0.40
PRKAG3 Q9UGI9 1/20 0.40
PRKAG2 Q9UGJ0 1/20 0.40
PRKAB1 Q9Y478 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA7 P36544 1/20 0.40
CHRNA4 P43681 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694458 0.89 CCR5 (0.53) CCR5CCL5CHRNB2CHRNB4CHRNA3
SCHEMBL4696366 0.89 CCR5 (0.46) KCNA5CCR5CCL5
SCHEMBL4694095 0.85 CCR5 (0.51) KCNA5CCR5CCL5
SCHEMBL4692349 0.83 CCR5 (0.54) CCR5CCL5
SCHEMBL4695293 0.83 CCR5 (0.46) ALDH1A1CCR5CCL5
SCHEMBL4695271 0.83 LMNA (0.53) CCR5CCL5CCR2
SCHEMBL4694257 0.83 CCR5 (0.48) CCR5CCL5
SCHEMBL4690556 0.81 CCR5 (0.51) CCR5CCL5
SCHEMBL4693578 0.80 CCR5 (0.53) ALDH1A1CCR5CCL5
SCHEMBL4693123 0.80 CCR5 (0.50) ALDH1A1CCR5CCL5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed