SCHEMBL4694458

SCHEMBL4694458

N[C@@H](CCN1CC2CN(C(=O)c3ccccc3)CC2C1)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 13/20 0.53
CHRNB2 P17787 1/20 0.50
CHRNB4 P30926 1/20 0.50
CHRNA3 P32297 1/20 0.50
CHRNA7 P36544 1/20 0.50
CHRNA4 P43681 1/20 0.50
CCL5 P13501 6/20 0.45
MAOB P27338 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694095 0.92 CCR5 (0.51) CCR5CCL5
SCHEMBL4690515 0.89 ALDH1A1 (0.47) CCR5CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL4695293 0.89 CCR5 (0.46) CCR5CCL5
SCHEMBL4694257 0.89 CCR5 (0.48) CCR5CCL5
SCHEMBL4695271 0.89 LMNA (0.53) CCR5CCL5
SCHEMBL4693284 0.89 CCR5 (0.53) CCR5CCL5
SCHEMBL4691929 0.89 CCR5 (0.48) CCR5CCL5
SCHEMBL3283162 0.89 CHRNB2 (0.54) CCR5CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL4693123 0.88 CCR5 (0.50) CCR5CCL5
SCHEMBL4691562 0.87 CHRM2 (0.46) CCR5CCL5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed