SCHEMBL4690600

SCHEMBL4690600

COc1cccc2c(C(N)=O)c(C(=O)N3CC4CN(CC[CH]c5ccccc5)C[C@H]4C3)[nH]c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
RECQL P46063 1/20 0.39
MCL1 Q07820 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ADRA1B P35368 2/20 0.38
HCRTR1 O43613 7/20 0.37
HCRTR2 O43614 7/20 0.37
TLR9 Q9NR96 1/20 0.36
TLR8 Q9NR97 1/20 0.36
TLR7 Q9NYK1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692504 0.77 HCRTR1 (0.44) MEN1KMT2AKDM4EALDH1A1GAA
SCHEMBL4690594 0.75 CCR5 (0.44) SMN1; SMN2KMT2AMAPTHCRTR1HCRTR2
SCHEMBL3290678 0.75 CCR5 (0.50) HCRTR1HCRTR2CCR5
SCHEMBL3285409 0.75 CCR5 (0.50) HCRTR1HCRTR2CCR5
SCHEMBL4690605 0.75 KDM4E (0.49) SMN1; SMN2MEN1KMT2AKDM4EALDH1A1
SCHEMBL4695880 0.74 CCR5 (0.40) HCRTR1HCRTR2CCR5
SCHEMBL4694094 0.74 CHRNB2 (0.44) SMN1; SMN2ALDH1A1GAAHPGDL3MBTL1
SCHEMBL4698176 0.74 CCR5 (0.40) HCRTR1HCRTR2CCR5
SCHEMBL4693258 0.74 HCRTR1 (0.41) KMT2APOLBGAAHCRTR1HCRTR2
SCHEMBL4694999 0.73 RECQL (0.40) SMN1; SMN2MEN1KMT2AALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed