SCHEMBL4690717

SCHEMBL4690717

NC(=O)C1[C@@H]2CN(C(=O)Cc3ccccc3)CC2CN1CC[CH]c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 2/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
KMT2A Q03164 1/20 0.38
ALDH1A1 P00352 4/20 0.37
TACR3 P29371 1/20 0.37
POLB P06746 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
TSHR P16473 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KDM4E B2RXH2 2/20 0.35
HSD11B1 P28845 1/20 0.34
GPR183 P32249 2/20 0.34
CCR5 P51681 1/20 0.34
LIPE Q05469 1/20 0.33
CACNA1G O43497 1/20 0.33
CACNA1H O95180 1/20 0.33
KCNH2 Q12809 1/20 0.33
GAA P10253 1/20 0.33
NPY5R Q15761 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692752 0.86 HTT (0.39) MEN1LMNAKMT2AALDH1A1POLB
SCHEMBL5232784 0.86 CHRNB2 (0.43) MEN1KMT2AALDH1A1SMN1; SMN2KCNH2
SCHEMBL5232761 0.85 CCR5 (0.35) LMNAALDH1A1KDM4ECCR5
SCHEMBL5235949 0.84 KMT2A (0.34) MEN1KMT2AALDH1A1TSHRSMN1; SMN2
SCHEMBL5235605 0.84 ALDH1A1 (0.36) ALDH1A1KDM4ECCR5GAA
SCHEMBL5229109 0.84 CHRNB2 (0.45) LMNAALDH1A1POLBTSHRSMN1; SMN2
SCHEMBL5237723 0.83 GRIN2B (0.39)
SCHEMBL5236454 0.83 GRIN2B (0.39)
SCHEMBL5235726 0.82 CCR5 (0.35) MEN1KMT2AALDH1A1KDM4EHSD11B1
SCHEMBL5232619 0.82 HSD11B1 (0.40) KMT2AALDH1A1KDM4EHSD11B1CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed