SCHEMBL4690983

SCHEMBL4690983

NC(=O)c1cccc(C2CC2)c1O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.49
MAPT P10636 2/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
HSD17B10 Q99714 1/20 0.44
PARP1 P09874 10/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
ADRA1A P35348 1/20 0.38
CXCR2 P25025 1/20 0.38
AURKA O14965 1/20 0.38
RPS6KB1 P23443 1/20 0.38
TAS1R3 Q7RTX0 2/20 0.38
TAS1R1 Q7RTX1 2/20 0.38
TAS1R2 Q8TE23 2/20 0.38
CNR1 P21554 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30100529 0.93 KDM4E (0.58) KDM4EMAPTMEN1KMT2AALDH1A1
SCHEMBL31465181 0.84 PARP1 (0.50) KDM4EMAPTMEN1KMT2AALDH1A1
SCHEMBL30689750 0.83 ALDH1A1 (0.50) KDM4EMEN1KMT2AALDH1A1HPGD
SCHEMBL1761171 0.82 KDM4E (0.38) KDM4EMAPTMEN1KMT2AALDH1A1
SCHEMBL1761183 0.82 KDM4E (0.38) KDM4EMAPTMEN1KMT2AALDH1A1
SCHEMBL1761170 0.82 KDM4E (0.38) KDM4EMAPTMEN1KMT2AALDH1A1
SCHEMBL6383642 0.82 ADRA1A (0.51) KDM4EMAPTMEN1KMT2AALDH1A1
SCHEMBL161548 0.82 ADRA1A (0.51) KDM4EMAPTMEN1KMT2AALDH1A1
SCHEMBL30666294 0.81 KDM4E (0.39) KDM4EMAPTMEN1KMT2AALDH1A1
Hydrochloric Acid SCHEMBL30170745 0.81 ADRA1A (0.50) KDM4EMAPTMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1521757-B1 TRICYCLIC SPIROPIPERIDINES OR SPIROPYRROLIDINES ASTRAZENECA AB (SE) 2008-01-30 EP disclosed