SCHEMBL4691592

SCHEMBL4691592

COc1ccc(-n2ncc(C(=O)N3CC4CN(CCCN)CC4C3)c2C(F)(F)F)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.41
PDK2 Q15119 1/20 0.41
HSD17B10 Q99714 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 3/20 0.39
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
ATM Q13315 1/20 0.39
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HCRTR1 O43613 2/20 0.38
HCRTR2 O43614 2/20 0.38
MAPK14 Q16539 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
PTPN1 P18031 1/20 0.38
HSD11B1 P28845 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691588 0.89 PDK1 (0.41) PDK1PDK2KDM4EALDH1A1MAPT
SCHEMBL4691935 0.85 KDM4E (0.42) PDK1PDK2KDM4EALDH1A1MAPT
SCHEMBL4693427 0.82 MAPT (0.42) ALDH1A1MAPTMEN1KMT2ALMNA
SCHEMBL4693420 0.78 MAPT (0.45) ALDH1A1MAPTKMT2ALMNAPOLB
SCHEMBL4691933 0.76 ALDH1A1 (0.42) PDK1PDK2KDM4EALDH1A1MAPT
SCHEMBL4691733 0.75 KMT2A (0.45) PDK1PDK2KDM4EALDH1A1MAPT
SCHEMBL4691829 0.75 KCNH2 (0.42)
SCHEMBL4689975 0.75 KDM4E (0.50) PDK1PDK2KDM4EALDH1A1MAPT
SCHEMBL4695680 0.74 CCR5 (0.45)
SCHEMBL4692260 0.74 PDK1 (0.45) PDK1PDK2KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed