SCHEMBL4691933

SCHEMBL4691933

NC(=O)Oc1ccc(-n2ncc(C(=O)N3CC4CN(CC[CH]c5ccccc5)C[C@H]4C3)c2C(F)(F)F)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
KDM4E B2RXH2 2/20 0.42
MAPT P10636 4/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
POLB P06746 1/20 0.41
LMNA P02545 3/20 0.38
HSD11B1 P28845 1/20 0.38
TDP1 Q9NUW8 2/20 0.38
PDK1 Q15118 1/20 0.36
PDK2 Q15119 1/20 0.36
MAPK11 Q15759 3/20 0.34
KMT2A Q03164 1/20 0.34
MET P08581 1/20 0.34
AXL P30530 1/20 0.34
MAPK14 Q16539 2/20 0.34
HCRTR1 O43613 2/20 0.33
HCRTR2 O43614 2/20 0.33
DDR1 Q08345 1/20 0.33
DDR2 Q16832 1/20 0.33
TMEM97 Q5BJF2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691732 0.90 KDM4E (0.43) ALDH1A1KDM4EMAPTSMN1; SMN2POLB
SCHEMBL4690551 0.88 MAPK14 (0.41) ALDH1A1SMN1; SMN2POLBLMNAMAPK11
SCHEMBL4691832 0.87 HCRTR1 (0.37) ALDH1A1KDM4EMAPTSMN1; SMN2POLB
SCHEMBL4692257 0.81 PDK1 (0.43) ALDH1A1KDM4EMAPTSMN1; SMN2POLB
SCHEMBL4694271 0.80 KDM4E (0.39) ALDH1A1KDM4EMAPTSMN1; SMN2POLB
SCHEMBL4690864 0.79 RIPK2 (0.40) MAPK11KMT2AMAPK14HCRTR1HCRTR2
SCHEMBL4689971 0.79 ALDH1A1 (0.44) ALDH1A1KDM4EMAPTSMN1; SMN2POLB
SCHEMBL4691588 0.78 PDK1 (0.41) ALDH1A1KDM4EMAPTSMN1; SMN2POLB
SCHEMBL4691935 0.77 KDM4E (0.42) ALDH1A1KDM4EMAPTSMN1; SMN2POLB
SCHEMBL4694244 0.77 EIF4A3 (0.45) ALDH1A1MAPTHSD11B1MAPK11MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed