SCHEMBL4691772

SCHEMBL4691772

N[C@@H](CCN1CC2CN(C(=O)c3ccccc3C(F)(F)F)CC2C1)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
HTR2B P41595 1/20 0.47
MAPK14 Q16539 1/20 0.47
CCR5 P51681 10/20 0.46
CCL5 P13501 4/20 0.42
RBP4 P02753 2/20 0.41
SCD O00767 2/20 0.40
MGLL Q99685 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4695175 0.85 CCR5 (0.47) CCR5CCL5RBP4
SCHEMBL4690615 0.84 HCRTR1 (0.52) CCR5CCL5MGLL
SCHEMBL4689905 0.83 CCR5 (0.52) CYP2C9CYP2C19HTR2BMAPK14CCR5
SCHEMBL4695158 0.83 CCR5 (0.55) CCR5CCL5
SCHEMBL4694458 0.81 CCR5 (0.53) CCR5CCL5
SCHEMBL4694311 0.81 CCL5 (0.44) CCR5CCL5
SCHEMBL4691786 0.81 HCRTR1 (0.52) CCR5CCL5
SCHEMBL4693261 0.80 HCRTR1 (0.51) CYP2C9CYP2C19MAPK14CCR5
SCHEMBL4691742 0.80 CCR5 (0.45) CCR5CCL5
SCHEMBL4690351 0.80 CCR5 (0.55) CCR5CCL5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed