SCHEMBL4691840

SCHEMBL4691840

COc1ccc(OC)c(C(=O)N2CC3CN(CCCNc4ccc(C)c(Cl)c4)CC3C2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.47
ALDH1A1 P00352 3/20 0.47
GFER P55789 1/20 0.47
LMNA P02545 2/20 0.43
HTT P42858 2/20 0.43
USP2 O75604 1/20 0.43
MCL1 Q07820 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
GAA P10253 2/20 0.41
MAPK1 P28482 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
HCRTR1 O43613 4/20 0.40
HCRTR2 O43614 4/20 0.40
POLB P06746 3/20 0.40
ABCB1 P08183 1/20 0.40
DUSP3 P51452 1/20 0.40
PTPN5 P54829 1/20 0.40
PTPN11 Q06124 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4695902 0.93 HCRTR2 (0.48) MAPTALDH1A1HTTGAAHCRTR1
SCHEMBL4691874 0.93 ALDH1A1 (0.43) MAPTALDH1A1LMNAGAACYP1A2
SCHEMBL4694353 0.92 KCNK3 (0.46) MAPTALDH1A1GFERLMNAHTT
SCHEMBL4690931 0.91 MAPT (0.51) MAPTALDH1A1LMNAHTTUSP2
SCHEMBL4694783 0.90 MAPT (0.46) MAPTALDH1A1LMNAHTTUSP2
SCHEMBL4691406 0.90 HCRTR1 (0.48) MAPTALDH1A1GAAHCRTR1HCRTR2
SCHEMBL4690310 0.89 MAPT (0.46) MAPTALDH1A1LMNAHTTUSP2
SCHEMBL4689521 0.88 MAPT (0.57) MAPTALDH1A1LMNAHTTUSP2
SCHEMBL4690506 0.88 HCRTR1 (0.52) MAPTALDH1A1LMNAGAAMAPK1
SCHEMBL4691831 0.87 MAPT (0.51) MAPTALDH1A1LMNASMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed