SCHEMBL4690551

SCHEMBL4690551

NC(=O)Oc1ccc(-n2ncc(C(=O)N3CC4CN(CC[CH]c5ccccc5)C[C@H]4C3)c2N)cc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 6/20 0.41
RIPK2 O43353 1/20 0.40
RAB9A P51151 4/20 0.39
LMNA P02545 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HPGD P15428 2/20 0.38
ALDH1A1 P00352 2/20 0.38
NPC1 O15118 2/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
PTGS1 P23219 1/20 0.38
LOX P28300 1/20 0.38
PTGS2 P35354 1/20 0.38
CA9 Q16790 1/20 0.38
PTPN1 P18031 1/20 0.36
POLB P06746 1/20 0.35
MAPK11 Q15759 2/20 0.35
BTK Q06187 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691933 0.88 ALDH1A1 (0.42) MAPK14LMNASMN1; SMN2ALDH1A1POLB
SCHEMBL4690142 0.86 MAPK14 (0.41) MAPK14RIPK2ALDH1A1
SCHEMBL4690864 0.82 RIPK2 (0.40) MAPK14RIPK2RAB9AHPGDNPC1
SCHEMBL4694466 0.81 RIPK2 (0.50) MAPK14RIPK2RAB9ALMNASMN1; SMN2
SCHEMBL4694244 0.80 EIF4A3 (0.45) MAPK14HPGDALDH1A1PTGS2MAPK11
SCHEMBL4693316 0.80 EIF4A3 (0.39) MAPK14RIPK2RAB9ALMNASMN1; SMN2
SCHEMBL4692885 0.79 MAPK14 (0.44) MAPK14RIPK2RAB9ALMNASMN1; SMN2
SCHEMBL4691732 0.78 KDM4E (0.43) MAPK14LMNASMN1; SMN2ALDH1A1POLB
SCHEMBL4693258 0.77 HCRTR1 (0.41) MAPK14LMNAPOLB
SCHEMBL4691832 0.77 HCRTR1 (0.37) LMNASMN1; SMN2ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed