SCHEMBL4692218

SCHEMBL4692218

Cc1ccc(NCCCN2CC3CN(C(=O)c4cccc(Cl)c4F)CC3C2)cc1Cl

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 8/20 0.42
MAPT P10636 4/20 0.41
ALDH1A1 P00352 4/20 0.41
HCRTR1 O43613 2/20 0.41
HCRTR2 O43614 2/20 0.41
GAA P10253 4/20 0.40
P2RX7 Q99572 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.39
PDE2A O00408 1/20 0.39
KDM4E B2RXH2 1/20 0.39
KCNK3 O14649 1/20 0.39
KCNK9 Q9NPC2 1/20 0.39
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
AGTR1 P30556 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694167 0.94 HCRTR1 (0.48) CCR5MAPTALDH1A1HCRTR1HCRTR2
SCHEMBL4691764 0.93 CCR5 (0.42) CCR5MAPTALDH1A1HCRTR1HCRTR2
SCHEMBL4694356 0.93 P2RX7 (0.43) CCR5MAPTALDH1A1GAAP2RX7
SCHEMBL4693334 0.92 ALDH1A1 (0.45) CCR5MAPTALDH1A1GAAP2RX7
SCHEMBL4691185 0.91 P2RX7 (0.43) CCR5MAPTALDH1A1HCRTR1HCRTR2
SCHEMBL4695648 0.91 HCRTR1 (0.48) CCR5MAPTALDH1A1HCRTR1HCRTR2
SCHEMBL4694387 0.91 GAA (0.41) CCR5MAPTALDH1A1HCRTR1HCRTR2
SCHEMBL4691872 0.91 HCRTR1 (0.47) CCR5MAPTALDH1A1HCRTR1HCRTR2
SCHEMBL4691905 0.91 HCRTR1 (0.47) CCR5MAPTALDH1A1HCRTR1HCRTR2
SCHEMBL4692676 0.91 P2RX7 (0.45) CCR5MAPTALDH1A1HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP disclosed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO disclosed