SCHEMBL4694356

SCHEMBL4694356

Cc1ccc(NCCCN2CC3CN(C(=O)c4cccc(Cl)c4Cl)CC3C2)cc1Cl

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 11/20 0.43
CCR5 P51681 3/20 0.42
ALDH1A1 P00352 4/20 0.41
MAPT P10636 2/20 0.41
KDM4E B2RXH2 2/20 0.39
GAA P10253 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692676 0.94 P2RX7 (0.45) P2RX7CCR5ALDH1A1MAPTKDM4E
SCHEMBL4691764 0.93 CCR5 (0.42) CCR5ALDH1A1MAPTKDM4EGAA
SCHEMBL4694387 0.93 GAA (0.41) P2RX7CCR5ALDH1A1MAPTKDM4E
SCHEMBL4692218 0.93 CCR5 (0.42) P2RX7CCR5ALDH1A1MAPTKDM4E
SCHEMBL4693334 0.92 ALDH1A1 (0.45) P2RX7CCR5ALDH1A1MAPTKDM4E
SCHEMBL4691872 0.91 HCRTR1 (0.47) CCR5ALDH1A1MAPTKDM4EGAA
SCHEMBL4692889 0.90 MAPT (0.45) CCR5ALDH1A1MAPTKDM4EGAA
SCHEMBL4694025 0.90 P2RX7 (0.48) P2RX7
SCHEMBL4693961 0.90 HCRTR1 (0.46) CCR5ALDH1A1MAPTKDM4EGAA
SCHEMBL3284097 0.89 CCR5 (0.41) CCR5ALDH1A1MAPTKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed