SCHEMBL4692628

SCHEMBL4692628

COc1cccc(C(=O)N2CC3CN(CCCNc4ccc(C)c(Cl)c4)CC3C2)c1OC

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.50
HCRTR2 O43614 2/20 0.50
ALDH1A1 P00352 6/20 0.45
KDM4E B2RXH2 4/20 0.45
LMNA P02545 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
HTT P42858 2/20 0.43
POLB P06746 1/20 0.43
HIF1A Q16665 1/20 0.42
CBX7 O95931 7/20 0.42
GAA P10253 1/20 0.42
HSD11B1 P28845 1/20 0.41
DRD3 P35462 1/20 0.41
SLC6A12 P48065 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691305 0.94 MAPT (0.42) HCRTR1HCRTR2ALDH1A1KDM4ELMNA
SCHEMBL4693956 0.92 HCRTR1 (0.49) HCRTR1HCRTR2ALDH1A1SMN1; SMN2NPC1
SCHEMBL4691406 0.92 HCRTR1 (0.48) HCRTR1HCRTR2ALDH1A1NPC1POLB
SCHEMBL4694080 0.91 HCRTR1 (0.40) HCRTR1HCRTR2ALDH1A1KDM4ESMN1; SMN2
SCHEMBL4693901 0.90 HCRTR1 (0.47) HCRTR1HCRTR2ALDH1A1KDM4ELMNA
SCHEMBL4694353 0.87 KCNK3 (0.46) HCRTR1HCRTR2ALDH1A1LMNASMN1; SMN2
SCHEMBL4691764 0.87 CCR5 (0.42) HCRTR1HCRTR2ALDH1A1KDM4ELMNA
SCHEMBL4692624 0.86 HCRTR1 (0.50) HCRTR1HCRTR2ALDH1A1KDM4ELMNA
SCHEMBL4690506 0.86 HCRTR1 (0.52) HCRTR1HCRTR2ALDH1A1LMNAGAA
SCHEMBL4691840 0.86 MAPT (0.47) HCRTR1HCRTR2ALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP disclosed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO disclosed